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TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50240899(cid_5280862 | 5,7-Dihydroxy-2-(4-hydroxy-phenyl)-3...)
Affinity DataIC50: 4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50292535(5,7-Dihydroxy-2-(4-hydroxy-phenyl)-3,6-dimethoxy-c...)
Affinity DataIC50: 50nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464571(CHEBI:70009 | Myricetin 3,3'',4''-Trimethylether |...)
Affinity DataIC50: 90nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50240898(CHEMBL161957 | 5,7-Dihydroxy-3,6-dimethoxy-2-(4-me...)
Affinity DataIC50: 220nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50140241(CHEBI:40279 | Allopurinol | Aloral | Aluline 100 |...)
Affinity DataIC50: 250nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355395(CHEMBL1834806)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355396(CHEMBL1834808)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355395(CHEMBL1834806)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355396(CHEMBL1834808)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355397(CHEMBL1834807)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355398(CHEMBL1834809)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355397(CHEMBL1834807)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355398(CHEMBL1834809)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355399(CHEMBL1834877)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355399(CHEMBL1834877)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464570(CHEMBL3407503)
Affinity DataIC50: 4.54E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355400(CHEMBL1834810)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50355401(CHEMBL1834811)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355400(CHEMBL1834810)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355401(CHEMBL1834811)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464572(CHEMBL3407749)
Affinity DataIC50: 6.95E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394654(CHEMBL188181)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464569(7-Trimethylkaempferol | CHEMBL77686)
Affinity DataIC50: 9.79E+3nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464573(CHEMBL521934)
Affinity DataIC50: 1.49E+4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394652(CHEMBL2165236)
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394653(CHEMBL2165235)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394655(CHEMBL2165237)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetXanthine dehydrogenase/oxidase(Bovine)
Universidad Nacional De C£Rdoba

Curated by ChEMBL
LigandPNGBDBM50464574(CHEMBL4294702)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of bovine milk xanthine oxidase using xanthine as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM26663((2S)-5,7-dihydroxy-8-(3-methylbut-2-en-1-yl)-2-phe...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
TBA

Curated by ChEMBL
LigandPNGBDBM50394656(CHEMBL2165240)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetNeuroepithelial cell-transforming gene 1 protein(Human)
Paris-Saclay University

Curated by ChEMBL
LigandPNGBDBM50366292(Dehydroroemerine)
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of Net1 (149 to 501 residues) (unknown origin) interaction with GDP-loaded His-tagged RhoA F25N mutant (1 to 180 residues) assessed as red...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetRho guanine nucleotide exchange factor 1(Human)
Paris-Saclay University

Curated by ChEMBL
LigandPNGBDBM50056922(cid_73677 | CHEMBL173530 | 1,4-Dihydroxy-10-methox...)
Affinity DataIC50: 1.87E+5nMAssay Description:Inhibition of p115 DHPH22 domain (395 to 766 residues) (unknown origin) interaction with GDP-loaded His-tagged RhoA F25N mutant (1 to 180 residues) a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi: <1nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022583(CHEMBL3298854)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022622(CHEMBL3299033)
Affinity DataKi:  5.90E+3nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022568(CHEMBL3298853)
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022568(CHEMBL3298853)
Affinity DataKi:  1.30E+4nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022567(CHEMBL3298852)
Affinity DataKi:  1.40E+4nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022567(CHEMBL3298852)
Affinity DataKi:  1.92E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022622(CHEMBL3299033)
Affinity DataKi:  1.94E+4nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM21447(4-(4-{[2-(4-chlorophenyl)phenyl]methyl}piperazin-1...)
Affinity DataKi:  2.08E+4nMAssay Description:Displacement of fluorescein-labeled BID from His-tagged MCL-1 (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022566(CHEMBL3298851)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022583(CHEMBL3298854)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetBcl-2-like protein 1(Human)
Institut De Chimie Des Substances Naturelles (Icsn)

Curated by ChEMBL
LigandPNGBDBM50022655(CHEMBL3299034)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of fluorescein-labeled BAK from His-tagged BCL-XL (unknown origin) after 1 hr by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed