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TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50025935(CHEMBL3144404 | {1-[1-(1-{2-[1-(Benzylamino-methyl...)
Affinity DataKi:  0.0260nMAssay Description:Compound was tested for inhibition of hog kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023090(Boc-Phe-His-Sta-Leu-4-amido-1-benzylpiperidine | C...)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023090(Boc-Phe-His-Sta-Leu-4-amido-1-benzylpiperidine | C...)
Affinity DataKi:  0.0640nMAssay Description:Inhibition of purified human kidney renin, fluorometric assay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50025934(CHEMBL3144405 | {1-[1-(1-{2-[1-(1-Benzyl-piperidin...)
Affinity DataKi:  0.0640nMAssay Description:Compound was tested for inhibition of human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023094(Boc-Phe-His-Sta-Leu-erythro-1,2-diphenyl-2-hydroxy...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023094(Boc-Phe-His-Sta-Leu-erythro-1,2-diphenyl-2-hydroxy...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023094(Boc-Phe-His-Sta-Leu-erythro-1,2-diphenyl-2-hydroxy...)
Affinity DataKi:  0.200nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077035(1-(1-{2-[4-Morpholin-4-yl-2-(2,2,2-trifluoro-ethox...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077032(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-(2,2,2-t...)
Affinity DataKi:  0.710nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077035(1-(1-{2-[4-Morpholin-4-yl-2-(2,2,2-trifluoro-ethox...)
Affinity DataKi:  0.860nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077041(1-(1-{2-[4-(1-Cyclopropylmethyl-piperidin-4-yloxy)...)
Affinity DataKi:  1nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50005463((R)-1H-Indole-2-carboxylic acid (1-methyl-2-oxo-5-...)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077041(1-(1-{2-[4-(1-Cyclopropylmethyl-piperidin-4-yloxy)...)
Affinity DataKi:  1.20nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM82387(CCK antagonist synthetic 22)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077032(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-(2,2,2-t...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077037(1-(1-{2-[4-(2-Morpholin-4-yl-ethoxy)-2-(2,2,2-trif...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023091(CHEMBL269752 | Iva-His-Pro-Phe-His-Sta-Leu-Phe-NH2)
Affinity DataKi:  1.5nMAssay Description:Inhibition of purified human kidney renin, fluorometric assay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077032(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-(2,2,2-t...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards rat liver Vasopressin V1a receptor by using functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019260(1H-Indole-2-carboxylic acid [5-(2-fluoro-phenyl)-2...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077037(1-(1-{2-[4-(2-Morpholin-4-yl-ethoxy)-2-(2,2,2-trif...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077039(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-trifluor...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077039(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-trifluor...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50025932(CHEMBL3144406 | Nitrate salt of {1-[1-(1-{2-[1-(1-...)
Affinity DataKi:  3.60nMAssay Description:Compound was tested for inhibition of human plasma reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077034(1-(1-{2-[2-(2,2,2-Trifluoro-ethoxy)-phenyl]-acetyl...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019252(1H-Indole-2-carboxylic acid (2-oxo-5-phenyl-2,3-di...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023050(CHEMBL40928 | {1-[1-(1-{2-[1-(1-Carbamoyl-2-phenyl...)
Affinity DataKi:  4.80nMAssay Description:Compound was tested for inhibition of human kidney reninMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023096(Boc-Phe-His-Sta-Leu-(+)-alpha-phenylthylamide | CH...)
Affinity DataKi:  6nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077034(1-(1-{2-[2-(2,2,2-Trifluoro-ethoxy)-phenyl]-acetyl...)
Affinity DataKi:  6nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rat)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  9.30nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077040(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-methoxy-...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023088(Boc-Phe-His-Sta-Leu-p-methoxybenzylamide | CHEMBL5...)
Affinity DataKi:  12nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023091(CHEMBL269752 | Iva-His-Pro-Phe-His-Sta-Leu-Phe-NH2)
Affinity DataKi:  17nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50016033(CHEMBL3085574 | {1-[1-{1-[2-(1-Benzylcarbamoyl-3-m...)
Affinity DataKi:  18nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023096(Boc-Phe-His-Sta-Leu-(+)-alpha-phenylthylamide | CH...)
Affinity DataKi:  19nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023091(CHEMBL269752 | Iva-His-Pro-Phe-His-Sta-Leu-Phe-NH2)
Affinity DataKi:  19nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50029649(1-(1-(4-(1-acetylpiperidin-4-yloxy)-2-methoxybenzo...)
Affinity DataKi:  19nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023092(Boc-Phe-His-Sta-Leu-(+)-1,2-diphenylthylamide | Bo...)
Affinity DataKi:  20nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50043194(1N-[7,7-dimethyl-1-spiro[2,3-dihydro-1H-indene-1,4...)
Affinity DataKi:  26nMAssay Description:Inhibition of radioligand [3H]-AVP binding to the vasopressin V2 receptor in rat kidney tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023092(Boc-Phe-His-Sta-Leu-(+)-1,2-diphenylthylamide | Bo...)
Affinity DataKi:  27nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023092(Boc-Phe-His-Sta-Leu-(+)-1,2-diphenylthylamide | Bo...)
Affinity DataKi:  28nMAssay Description:Inhibition of hog kidney renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023092(Boc-Phe-His-Sta-Leu-(+)-1,2-diphenylthylamide | Bo...)
Affinity DataKi:  29nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using the natural substrate partially pure angiotensinogen at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077038(1-{1-[2-(2,4-Dimethoxy-phenyl)-acetyl]-piperidin-4...)
Affinity DataKi:  33nMAssay Description:Binding affinity for human oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023092(Boc-Phe-His-Sta-Leu-(+)-1,2-diphenylthylamide | Bo...)
Affinity DataKi:  36nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023087(Boc-Phe-His-Sta-Leu-Phe-NH2 | Boc-Phe-His-Sta-Leu-...)
Affinity DataKi:  36nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023087(Boc-Phe-His-Sta-Leu-Phe-NH2 | Boc-Phe-His-Sta-Leu-...)
Affinity DataKi:  36nMAssay Description:Inhibition of human plasma renin at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50077040(1-(1-{2-[4-(1-Acetyl-piperidin-4-yloxy)-2-methoxy-...)
Affinity DataKi:  36nMAssay Description:Binding affinity for rat uterine oxytocin receptor (rOTr)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50023086(Boc-Phe-His-Sta-Leu-1-hydroxy-1-phenyl-2-propylami...)
Affinity DataKi:  36nMAssay Description:Inhibition of purified human kidney renin, radioimmunoassay using a synthetic tetradecapeptide renin substrate at 10e-9 M concentrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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