Affinity DataIC50: 1nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 126nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Antagonist activity at FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated degranulation after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 251nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonistic activity against P2X7 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 631nMAssay Description:In vitro antagonism of P2X 7 receptor in THP-1 (human pre-monocytic) cells.More data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Intrinsic activity at FPR1 in human neutrophils assessed as increase in calcium mobilization by FLIPR assay relative to fMLFMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human FPR1 in human neutrophils assessed as inhibition of fMLF-stimulated intracellular calcium mobilisation by FLIPR assayMore data for this Ligand-Target Pair
