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Report error Found 218 with Last Name = 'fattori' and Initial = 'r'
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM50219407(CHEMBL84350)
Affinity DataKi:  5nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataKi:  38nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM50219414(CHEMBL79661)
Affinity DataKi:  60nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219411(CHEMBL82934)
Affinity DataKi:  63nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219417(CHEMBL421343)
Affinity DataKi:  128nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219409(CHEMBL354743)
Affinity DataKi:  138nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataKi:  149nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219404(CHEMBL79739)
Affinity DataKi:  199nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219406(CHEMBL309420)
Affinity DataKi:  208nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219413(CHEMBL81226)
Affinity DataKi:  212nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219405(CHEMBL81020)
Affinity DataKi:  235nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219410(CHEMBL311025)
Affinity DataKi:  237nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219408(CHEMBL84115)
Affinity DataKi:  397nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219416(CHEMBL167389)
Affinity DataKi:  473nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219412(CHEMBL82882)
Affinity DataKi:  498nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236453(CHEMBL4068323)
Affinity DataKi:  2.30E+3nMAssay Description:Inhibitory activity against beta-glucosidase of sweet almondMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236360(CHEMBL4066708)
Affinity DataKi:  4.30E+4nMAssay Description:Non-competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated fo...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236359(CHEMBL4086085)
Affinity DataKi:  4.84E+4nMAssay Description:Competitive inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using H3K4me1 peptide as substrate preincubated for 15...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540648(CHEMBL4639944)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540643(CHEMBL4639941)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540639(CHEMBL4632810)
Affinity DataIC50:  0.130nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540640(CHEMBL4641768)
Affinity DataIC50:  0.140nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540649(CHEMBL4642214)
Affinity DataIC50:  0.160nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540655(CHEMBL4635889)
Affinity DataIC50:  0.170nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540642(CHEMBL4649085)
Affinity DataIC50:  0.180nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540644(CHEMBL4639413)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540638(CHEMBL4649563)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540645(CHEMBL4645937)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540646(CHEMBL4634153)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540654(CHEMBL4642738)
Affinity DataIC50:  0.270nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540653(CHEMBL4637660)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540641(CHEMBL4636234)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540651(CHEMBL4645131)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540652(CHEMBL4638582)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540647(CHEMBL4641915)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50155773(CHEMBL3781751 | US9469597, 5)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Human)
European Institute of Oncology Irccs

Curated by ChEMBL
LigandPNGBDBM50540650(CHEMBL4640188)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human LSD1 expressed in Escherichia coli using biotinylated H3K4me as substrate by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM254603(US10214477, Example 5 | US9469597, 4 | US9670136, ...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using biotinylated H3K4me1 peptide as substrate preincubated for 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM50219407(CHEMBL84350)
Affinity DataIC50:  2nMAssay Description:Inhibition of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236447(CHEMBL4069817)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236444(CHEMBL4090812)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236441(CHEMBL4072541)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219418(CHEMBL450274)
Affinity DataIC50:  12nMAssay Description:Inhibition of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236456(CHEMBL4081995)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
LigandPNGBDBM50219414(CHEMBL79661)
Affinity DataIC50:  21nMAssay Description:Inhibition of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A/REST corepressor 1(Human)
European Institute of Oncology

Curated by ChEMBL
LigandPNGBDBM50236457(CHEMBL4074211)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using [Lys(Me1)4]-Histone H3 (1 to 21 residues)-GGK(biotin) as sub...More data for this Ligand-Target Pair
LigandPNGBDBM50219412(CHEMBL82882)
Affinity DataIC50:  25nMAssay Description:Inhibition of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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