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TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476613(CHEMBL233309)
Affinity DataEC50:  25nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476614(CHEMBL392421)
Affinity DataEC50:  9.80nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476617(CHEMBL391350)
Affinity DataEC50:  13nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476611(CHEMBL233729)
Affinity DataEC50:  11nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476620(CHEMBL231872)
Affinity DataEC50:  46nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476619(CHEMBL394406)
Affinity DataEC50:  52nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476622(CHEMBL233517)
Affinity DataEC50:  155nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476624(CHEMBL233516)
Affinity DataEC50:  16nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476626(CHEMBL395221)
Affinity DataEC50:  32nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476627(CHEMBL233308)
Affinity DataEC50:  3.5nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476625(CHEMBL233740)
Affinity DataEC50:  339nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476621(CHEMBL394408)
Affinity DataEC50:  46nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476616(CHEMBL233311)
Affinity DataEC50:  120nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476628(CHEMBL392422)
Affinity DataEC50:  17nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476615(CHEMBL233310)
Affinity DataEC50:  65nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataEC50:  0.0794nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1C(African clawed frog)
University College London

Curated by ChEMBL
LigandPNGBDBM50476612(CHEMBL233728)
Affinity DataEC50:  3.30nMAssay Description:Effect on pigment aggregation in Xenopus laevis melanophoresMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50020882(CHEMBL103623 | 1-(4,4-Diphenyl-but-3-enyl)-1,2,5,6...)
Affinity DataIC50: 200nMAssay Description:Binding affinity to GAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 1(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50003634(1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxyli...)
Affinity DataIC50: 200nMAssay Description:Binding affinity to GAT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50039246((S)-1-(2-(tris(4-methoxyphenyl)methoxy)ethyl)piper...)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to GAT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50003624(Nipecotic | Piperidine-3-carboxylic acid(nipecotic...)
Affinity DataIC50: 6.60E+4nMAssay Description:Binding affinity to GAT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 2(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 6.60E+4nMAssay Description:Binding affinity to GAT2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM50003624(Nipecotic | Piperidine-3-carboxylic acid(nipecotic...)
Affinity DataIC50: 1.10E+5nMAssay Description:Binding affinity to GAT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetSodium- and chloride-dependent GABA transporter 3(Human)
Zentrum F£R Pharmaforschung

Curated by ChEMBL
LigandPNGBDBM90787(SMR000326834 | cid_11957555 | GUVACINE | MLS000859...)
Affinity DataIC50: 1.10E+5nMAssay Description:Binding affinity to GAT3More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2010
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086013(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.0500nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086033(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086017(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086004(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086032(N-[2-(2-Methoxy-6H-isoindolo[2,1-a]indol-11-yl)-et...)
Affinity DataKi:  0.170nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086029(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086020(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.210nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086028(N-[2-(2-Ethoxy-6H-isoindolo[2,1-a]indol-11-yl)-eth...)
Affinity DataKi:  0.260nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.263nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.339nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476627(CHEMBL233308)
Affinity DataKi:  0.355nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086001(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086005(N-[2-(10-Methoxy-5,6-dihydro-indolo[2,1-a]isoquino...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476611(CHEMBL233729)
Affinity DataKi:  0.537nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1A expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476612(CHEMBL233728)
Affinity DataKi:  0.676nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476617(CHEMBL391350)
Affinity DataKi:  0.676nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086011(Cyclopropanecarboxylic acid [2-(2-methoxy-6H-isoin...)
Affinity DataKi:  0.950nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476626(CHEMBL395221)
Affinity DataKi:  1.10nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476628(CHEMBL392422)
Affinity DataKi:  1.30nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476613(CHEMBL233309)
Affinity DataKi:  1.30nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50086025(N-[2-(11-Methoxy-6,7-dihydro-5H-benzo[3,4]azepino[...)
Affinity DataKi:  1.41nMAssay Description:Binding affinity towards recombinant human melatonin receptor type 1B expressed in NIH 3T3 cells using 2-[121I]iodomelatonin radioligand binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/25/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476614(CHEMBL392421)
Affinity DataKi:  1.5nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Human)
King'S College London

Curated by ChEMBL
LigandPNGBDBM50476620(CHEMBL231872)
Affinity DataKi:  1.70nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT2 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
TargetMelatonin receptor type 1A(Human)
University College London

Curated by ChEMBL
LigandPNGBDBM50476626(CHEMBL395221)
Affinity DataKi:  1.80nMAssay Description:Displacement of 2[125I]iodomelatonin from human recombinant MT1 receptor expressed in NIH3T3 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2020
Entry Details Article
PubMed
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