Compile Data Set for Download or QSAR
Report error Found 505 with Last Name = 'fernández-ruiz' and Initial = 'j'
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50265621(HU-308 | ((1R,4S,5R)-4-(2,6-dimethoxy-4-(2-methylo...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532456(CHEMBL4581919)
Affinity DataEC50:  299nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532474(CHEMBL4465748)
Affinity DataEC50:  191nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532440(CHEMBL4585657)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50265621(HU-308 | ((1R,4S,5R)-4-(2,6-dimethoxy-4-(2-methylo...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21281(WIN55212-2 | CHEMBL188 | (2,3-dihydro-5-methyl-3-(...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532474(CHEMBL4465748)
Affinity DataEC50:  191nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532456(CHEMBL4581919)
Affinity DataEC50:  299nMAssay Description:Agonist activity at human CB1 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532455(CHEMBL4557358)
Affinity DataEC50:  95nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as induction of [35S]-GTPgammaS binding after 60 mins by liquid sc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50405853(CHEMBL5273189)
Affinity DataEC50:  900nMAssay Description:Inverse agonist activity at human GPR55 expressed in HEK293 cells coexpressing serum response element assessed as reduction in MAPK/ERK signalling pa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2024
Entry Details
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156102(CHEMBL3781953)
Affinity DataEC50:  392nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells after 30 mins by [35S]-GTPgammaS binding assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156103(CHEMBL3781521)
Affinity DataEC50:  22nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156104(CHEMBL3780020)
Affinity DataEC50:  25nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156105(CHEMBL3781437)
Affinity DataEC50:  25nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156106(CHEMBL3779954)
Affinity DataEC50:  18nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156102(CHEMBL3781953)
Affinity DataEC50:  8.20nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156116(CHEMBL3781224)
Affinity DataEC50:  29nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156107(CHEMBL3779969)
Affinity DataEC50:  16nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156108(CHEMBL3781158)
Affinity DataEC50:  20nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156119(CHEMBL3781764)
Affinity DataEC50:  20nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156109(CHEMBL3781297)
Affinity DataEC50:  27nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156110(CHEMBL3780529)
Affinity DataEC50:  30nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156112(CHEMBL3780748)
Affinity DataEC50:  28nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156114(CHEMBL3781085)
Affinity DataEC50:  32nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156115(CHEMBL3781210)
Affinity DataEC50:  28nMAssay Description:Antagonist activity at recombinant human GPR55 expressed in HEK293 cells assessed as inhibition of LPI mediated receptor activation by measuring LPI ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156120(CHEMBL3780056)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156103(CHEMBL3781521)
Affinity DataEC50:  0.690nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156104(CHEMBL3780020)
Affinity DataEC50:  8.70nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156105(CHEMBL3781437)
Affinity DataEC50:  0.400nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156106(CHEMBL3779954)
Affinity DataEC50:  1.30nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156102(CHEMBL3781953)
Affinity DataEC50:  0.510nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156107(CHEMBL3779969)
Affinity DataEC50:  0.600nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156108(CHEMBL3781158)
Affinity DataEC50:  0.880nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetG-protein coupled receptor 55(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50156112(CHEMBL3780748)
Affinity DataEC50:  6.40nMAssay Description:Partial agonist activity at recombinant human GPR55 expressed in HEK293 cells after 5 mins by xCELLigence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2017
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataIC50: 4.20nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532442(CHEMBL4444725)
Affinity DataIC50: 4.20nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 8.30nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50072775(ChEMBL_75020 | 5-(1,1-Dimethyl-heptyl)-2-[(1R,2R,5...)
Affinity DataIC50: 8.30nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCannabinoid receptor 1(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM21278(SR141716 | 5-(4-chlorophenyl)-1-(2,4-dichloropheny...)
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO cell membranes assessed as reduction in GTPgammaS binding after 30 mins by microbeta count...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataIC50: 14nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
IQM-CSIC

Curated by ChEMBL
LigandPNGBDBM50532454(CHEMBL4588694)
Affinity DataIC50: 14nMAssay Description:Agonist activity at human CB2 receptor expressed in HEK293 cell membranes assessed as inhibition of forskolin-stimulated cAMP accumulation after 60 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/27/2021
Entry Details Article
PubMed
Displayed 1 to 50 (of 505 total ) | Next | Last >>
Jump to: