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TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246899((S)-2-(3-((S)-1-carboxy-5-(4-iodobenzamido)pentyl)...)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)
Affinity DataKi:  0.194nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246934((S)-2-(3-((S)-1-carboxy-5-(4-fluorobenzamido)penty...)
Affinity DataKi:  0.256nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246935((S)-2-(3-((S)-1-carboxy-5-(3-iodonicotinamido)pent...)
Affinity DataKi:  0.351nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50246935((S)-2-(3-((S)-1-carboxy-5-(3-iodonicotinamido)pent...)
Affinity DataKi:  0.557nMAssay Description:Inhibition of PSMA in human LNCaP cell extract using [3H]NAAG by fluorescence-based assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304738(2-(3-((S)-1-carboxy-3-methylbutyl)ureido)pentanedi...)
Affinity DataKi:  0.75nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304722((S)-2-(3-((S)-1-Carboxybut-3-ynyl)ureido)-6-(4-iod...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304731((S)-2-(3-((S)-1-Carboxy-2-(furan-2-yl)ethyl)ureido...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304751((S)-2-(3-((S)-1-Carboxybut-3-enyl)ureido)-6-(4-iod...)
Affinity DataKi:  11nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304735((S)-2-(3-((S)-1-Carboxy-2-(thiazol-4-yl)ethyl)urei...)
Affinity DataKi:  16.1nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304732((S)-2-(3-((S)-1-Carboxy-2-(thiophen-2-yl)ethyl)ure...)
Affinity DataKi:  16.2nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304727((S)-2-(3-((S)-1-Carboxy-3-(methylthio)propyl)ureid...)
Affinity DataKi:  23nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304728((S)-2-(3-((S)-4-(Acetylthio)-1-carboxybutyl)ureido...)
Affinity DataKi:  24.1nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304723((S)-2-(3-((S)-1-Carboxybutyl)ureido)-6-(4-iodobenz...)
Affinity DataKi:  52.3nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304715(2-(4-Hydroxy-3-methoxyphenyl)-2-(3-((S)-1-isopropo...)
Affinity DataKi:  81nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304729((S)-2-(3-((S)-Carboxy(4-hydroxyphenyl)methyl)ureid...)
Affinity DataKi:  85.1nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304737((S)-2-(3-((S)-1-carboxy-2-(pyridin-3-yl)ethyl)urei...)
Affinity DataKi:  97.2nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304736((S)-2-(3-((S)-1-Carboxy-2-(pyridin-4-yl)ethyl)urei...)
Affinity DataKi:  105nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304725((S)-2-(3-((S)-1-Carboxy-2-cyanoethyl)ureido)-6-(4-...)
Affinity DataKi:  132nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304714(2-(4-Hydroxy-3-methoxyphenyl)-2-(3-((S)-1-methoxy-...)
Affinity DataKi:  153nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304713((S)-2-(3-(Carboxy(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataKi:  250nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304724((2S)-2-(3-((1S)-1-carboxy-2-(oxiran-2-yl)ethyl)ure...)
Affinity DataKi:  254nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304717(2-(4-Hydroxy-3-iodophenyl)-2-(3-((S)-1-isopropoxy-...)
Affinity DataKi:  275nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304730((S)-2-(3-(Carboxy(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataKi:  285nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304750((S)-1-(3-(1-Carboxy-5-(4-iodobenzamido)pentyl)urei...)
Affinity DataKi:  318nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304726((S)-2-(3-((S)-3-Amino-1-carboxy-3-oxopropyl)ureido...)
Affinity DataKi:  320nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304718((S)-2-(3-bromo-4-hydroxyphenyl)-2-(3-((S)-1-methox...)
Affinity DataKi:  400nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304716((S)-2-(4-Hydroxy-3-iodophenyl)-2-(3-((S)-1-methoxy...)
Affinity DataKi:  475nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304719((S)-2-(3,5-dibromo-4-hydroxyphenyl)-2-(3-((S)-1-me...)
Affinity DataKi:  575nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304739(2-(3-(1-Carboxy-2-(4-hydroxyphenyl)ethyl)ureido)-4...)
Affinity DataKi:  700nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304711((S)-2-(3-((S)-carboxy(4-hydroxyphenyl)methyl)ureid...)
Affinity DataKi:  775nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304733((S)-2-(3-((R)-1-Carboxy-2-(furan-2-yl)ethyl)ureido...)
Affinity DataKi:  794nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304734((S)-2-(3-((R)-1-Carboxy-2-(thiophen-2-yl)ethyl)ure...)
Affinity DataKi:  795nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304748((S)-2-(3-(Carboxymethyl)ureido)-6-(4-iodobenzamido...)
Affinity DataKi:  1.32E+3nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304720((S)-2-(3-Fluoro-4-hydroxyphenyl)-2-(3-(1-methoxy-4...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304742((S)-3-(2-Carboxy-2-(3-(1-carboxy-3-methylbutyl)ure...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304749((S)-2-(3-(3-Carboxypropyl)ureido)-6-(4-iodobenzami...)
Affinity DataKi:  3.43E+3nMAssay Description:Inhibition of human cloned glutamate carboxypeptidase 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304744((S)-2-(3-((S)-1-Carboxy-3-(methylthio)propyl)ureid...)
Affinity DataKi:  3.50E+3nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304746((S)-5-amino-2-(3-((S)-1-methoxy-4-methyl-1-oxopent...)
Affinity DataKi:  7.50E+3nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304740(2-(3-(1-Carboxy-2-(4-hydroxy-3-iodophenyl)ethyl)ur...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304712((2S)-2-(3-(carboxy(3,5-dihydroxyphenyl)methyl)urei...)
Affinity DataKi:  1.30E+4nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304710((S)-2-(3-(Carboxy(3-hydroxyphenyl)methyl)ureido)-4...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304747((S)-2-(3-((S)-1-Carboxy-2-(1H-indol-3-yl)ethyl)ure...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304709((S)-2-(3-hydroxyphenyl)-2-(3-(1-methoxy-4-methyl-1...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304743((S)-3-(2-Carboxy-2-(3-(1-methoxy-4-methyl-1-oxopen...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304721((S)-2-(4-Fluoro-3-methoxyphenyl)-2-(3-(1-methoxy-4...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304741((S)-3-(3-Hydroxyphenyl)-2-(3-(1-methoxy-4-methyl-1...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate carboxypeptidase 2(Human)
Institutions

Curated by ChEMBL
LigandPNGBDBM50304745((S)-2-(3-((S)-1-Methoxy-4-methyl-1-oxopentan-2-yl)...)
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of glutamate carboxypeptidase 2 in human LNCaP cells by fluorescence based NAALADase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Human)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50268077((S)-4-(2-hydroxy-3-(1-(4-methoxyphenyl)-2-methylpr...)
Affinity DataIC50:  0.00130nMAssay Description:Inhibition of beta2 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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