TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 0.0940nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1A adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1A adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1A adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1A adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1B adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor serotonergic receptor in human HeLa cellsMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1D adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor serotonergic receptor in human HeLa cellsMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1A adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor serotonergic receptor in human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1D adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1B adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1D adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1D adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1B adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human CA12 by stopped-flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Inhibition of [3H]-8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor serotonergic receptor in human HeLa cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.90nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.10nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Inhibition of human CA2 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Università degli Studi di Torino
Curated by ChEMBL
Università degli Studi di Torino
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Inhibition of [3H]-prazosin binding to cloned human Alpha-1B adrenergic receptor in CHO-cells (chinese hamster ovary cells)More data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 6.60nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition of human CA9 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.10nMAssay Description:Inhibition of human CA12 by CO2 hydration activity based stopped flow assayMore data for this Ligand-Target Pair
