TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.0726nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0900nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.0978nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.101nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.106nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.137nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Displacement of [3H]PK11195 from rat PBR receptorMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor alpha (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.231nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.240nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.242nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.242nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.253nMAssay Description:Displacement of [3H]nociceptin from human recombinant NOP receptor expressed in CHO cells after 60 mins by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.299nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.370nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.370nMAssay Description:Displacement of [11C]PBR28 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.510nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.680nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.730nMAssay Description:Binding affinity to PBR in Sprague-Dawley rat mitochondrial tissueMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 0.970nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 0.997nMAssay Description:Displacement of [3H]PK11195 from human PBR receptorMore data for this Ligand-Target Pair
TargetGABA A receptor alpha-1/beta-1/gamma-2(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to GABA alpha-1-beta-1-gamma-2 receptorMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-6/beta-2/gamma-2(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: >1nMAssay Description:Binding affinity to GABA alpha-6-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.07nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 1.09nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Displacement of [11C]PBR28 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 1.51nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.57nMAssay Description:Displacement of [11C]PK11195 from high affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 1.82nMAssay Description:Displacement of [11C]PK11195 from mixed affinity binding site of TSPO in human brain membrane homogenate by scintillation countingMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 1.84nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 2.17nMAssay Description:Displacement of [125I]T3 from recombinant thyroid hormone receptor beta (unknown origin) expressed in sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 2.5nMAssay Description:Binding affinity to PBR in human mitochondrial tissueMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 2.51nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 2.92nMAssay Description:Displacement of [11C]PK11195 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 2.95nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine His-tagged human recombinant TRbeta1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Metabasis Therapeutics Inc
Curated by ChEMBL
Metabasis Therapeutics Inc
Curated by ChEMBL
Affinity DataKi: 3.74nMAssay Description:Displacement of [125I]3,5,3'-triiodo-L-thyronine from His-tagged human recombinant TRalpha1 by scintillation proximity assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute of Mental Health
Curated by ChEMBL
National Institute of Mental Health
Curated by ChEMBL
Affinity DataKi: 4.28nMAssay Description:Displacement of [11C]PBR28 from TSPO in rat kidney mitochondrial membraneMore data for this Ligand-Target Pair
