Compile Data Set for Download or QSAR
Found 262 with Last Name = 'gilmer' and Initial = 'jf'
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303940(2-(Benzylaminocarbonyloxy-)5-O-Salicyloyl-1,4:3,6-...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350604(CHEMBL1812922)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350604(CHEMBL1812922)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303950(CHEMBL583687 | Isosorbide-2-benzylcarbamate-5-(o-t...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350606(CHEMBL1812924)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350607(CHEMBL1812925)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350623(CHEMBL1812941)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350606(CHEMBL1812924)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350623(CHEMBL1812941)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50253229(CHEMBL445695 | Isosorbide-2-(benzylcarbamate)-5-mo...)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of human plasma BuchE after 60 mins by carbamylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388945(CHEMBL2063430)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-2 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50253231((3R,3aR,6S,6aR)-6-(benzylcarbamoyloxy)hexahydrofur...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of human plasma BuchE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50253231((3R,3aR,6S,6aR)-6-(benzylcarbamoyloxy)hexahydrofur...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350599(CHEMBL1812914)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50252786(CHEMBL492635 | Isosorbide-2-benzylcarbamate-5-cycl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human plasma BuchE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388949(CHEMBL2063518)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-9 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303952(2-(Dimethylaminocarbonyloxy-)5-O-Salicyloyl-1,4:3,...)
Affinity DataIC50:  6.40nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388952(CHEMBL2063432)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-2 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350607(CHEMBL1812925)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388952(CHEMBL2063432)
Affinity DataIC50:  8.10nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-9 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350603(CHEMBL1812921)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303951(2-(Ethylaminocarbonyloxy-)5-O-Salicyloyl-1,4:3,6-d...)
Affinity DataIC50:  9.60nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350613(CHEMBL1812931)
Affinity DataIC50:  9.80nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388951(CHEMBL2063433)
Affinity DataIC50:  10nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-2 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350599(CHEMBL1812914)
Affinity DataIC50:  10nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50424987(CHEMBL2311774)
Affinity DataIC50:  11nMAssay Description:Inhibition of human recombinant MMP-13 after 45 mins by fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50253266((3R,3aR,6S,6aR)-6-(benzylcarbamoyloxy)hexahydrofur...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human plasma BuchE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388951(CHEMBL2063433)
Affinity DataIC50:  12nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-9 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50253266((3R,3aR,6S,6aR)-6-(benzylcarbamoyloxy)hexahydrofur...)
Affinity DataIC50:  12nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350611(CHEMBL1812929)
Affinity DataIC50:  13nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350611(CHEMBL1812929)
Affinity DataIC50:  13nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350615(CHEMBL1812933)
Affinity DataIC50:  13nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50424995(CHEMBL2311772)
Affinity DataIC50:  13nMAssay Description:Inhibition of human recombinant MMP-9 after 45 mins by fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350602(CHEMBL1812920)
Affinity DataIC50:  14nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350615(CHEMBL1812933)
Affinity DataIC50:  14nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350600(CHEMBL1812915)
Affinity DataIC50:  15nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50388949(CHEMBL2063518)
Affinity DataIC50:  15nMAssay Description:Inhibition of p-aminophenylmercuric acetate stimulated human recombinant MMP-2 using (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrop...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350594(CHEMBL1812961)
Affinity DataIC50:  15nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303941(2-(Benzylaminocarbonyloxy-)5-O-(m-hydroxybenzoyl)-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350603(CHEMBL1812921)
Affinity DataIC50:  16nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350602(CHEMBL1812920)
Affinity DataIC50:  16nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350612(CHEMBL1812930)
Affinity DataIC50:  16nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50303943(2-(Benzylaminocarbonyloxy-)5-O-(o-nitro-benzoyl)-1...)
Affinity DataIC50:  18nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350612(CHEMBL1812930)
Affinity DataIC50:  19nMAssay Description:Inhibition of AMPA-activated human recombinant MMP9 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50004000((3aS,8aR)-1,3a,8-trimethyl-1,2,3,3a,8,8a-hexahydro...)
Affinity DataIC50:  19nMAssay Description:Inhibition of BuChE in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350594(CHEMBL1812961)
Affinity DataIC50:  20nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50424995(CHEMBL2311772)
Affinity DataIC50:  21nMAssay Description:Inhibition of human recombinant MMP-2 after 45 mins by fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350605(CHEMBL1812923)
Affinity DataIC50:  22nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50350632(CHEMBL1812950)
Affinity DataIC50:  23nMAssay Description:Inhibition of AMPA-activated human recombinant MMP2 using fluorogenic substrate (7-methoxycoumarin-4-yl)-acetyl-pro-Leu-Gly-Leu-(3-(2,4-dinitrophenyl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCollagenase 3(Homo sapiens (Human))
Trinity College

Curated by ChEMBL
LigandPNGBDBM50424985(CHEMBL2311776)
Affinity DataIC50:  23nMAssay Description:Inhibition of human recombinant MMP-13 after 45 mins by fluorogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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