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TargetHistone deacetylase 2(Human)
Wroclaw University

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant HDAC2 expressed in baculovirus using AMC-K(Ac)GL as substrate by microplate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMetallo-beta-lactamase type 2(Pseudomonas aeruginosa (g-Proteobacteria))
Wroclaw University

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  380nMAssay Description:Inhibition of bacterial New Delhi metallo-beta-lactamase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetThioredoxin reductase(Escherichia coli (strain K12))
Wroclaw University

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataKi:  520nMAssay Description:Competitive inhibition of Escherichia coli TrxR assessed as inhibition constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetToxin B(Peptoclostridium difficile)
Wroclaw University

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of Clostridium difficile full length Toxin BMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197353(CHEMBL3932329)
Affinity DataIC50:  121nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197347(Ebselen Diselenide)
Affinity DataIC50:  230nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetReplicase polyprotein 1ab(2019-nCoV)
University Ofamsterdam

LigandPNGBDBM50197301(CHEMBL3922662 | ebselen derivative 1d)
Affinity DataIC50:  236nMAssay Description:The inhibitor was screened against recombinant PL​pro​SARS and PL​pro​CoV2 at 37°Cin the assay buffer as described above. For...More data for this Ligand-Target Pair
In DepthDetails

TargetReplicase polyprotein 1ab(2019-nCoV)
University Ofamsterdam

LigandPNGBDBM50197349(CHEMBL3983492 | ebselen derivative 1e)
Affinity DataIC50:  256nMAssay Description:The inhibitor was screened against recombinant PL​pro​SARS and PL​pro​CoV2 at 37°Cin the assay buffer as described above. For...More data for this Ligand-Target Pair
In DepthDetails

TargetReplicase polyprotein 1ab(2019-nCoV)
University Ofamsterdam

LigandPNGBDBM50197300(CHEMBL3912164 | ebselen derivative 2e)
Affinity DataIC50:  263nMAssay Description:The inhibitor was screened against recombinant PL​pro​SARS and PL​pro​CoV2 at 37°Cin the assay buffer as described above. For...More data for this Ligand-Target Pair
In DepthDetails

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197302(CHEMBL3920474)
Affinity DataIC50:  320nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetReplicase polyprotein 1ab(2019-nCoV)
University Ofamsterdam

LigandPNGBDBM50197297(CHEMBL3928799 | ebselen derivative 2d)
Affinity DataIC50:  339nMAssay Description:The inhibitor was screened against recombinant PL​pro​SARS and PL​pro​CoV2 at 37°Cin the assay buffer as described above. For...More data for this Ligand-Target Pair
In DepthDetails

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197323(CHEMBL3931605)
Affinity DataIC50:  920nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197348(CHEMBL3940631)
Affinity DataIC50:  935nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197313(CHEMBL3930560)
Affinity DataIC50:  1.35E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197299(CHEMBL3913676)
Affinity DataIC50:  2.07E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197303(CHEMBL3892953)
Affinity DataIC50:  2.35E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM34233(2-Phenyl-benzo[d]isoselenazol-3-one | 2-Phenyl-ben...)
Affinity DataIC50:  2.43E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197304(CHEMBL3913688)
Affinity DataIC50:  2.67E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197352(CHEMBL3912588)
Affinity DataIC50:  3.43E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197344(CHEMBL3903564)
Affinity DataIC50:  4.47E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM106944(US8592468, EbSe2)
Affinity DataIC50:  4.97E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197297(CHEMBL3928799 | ebselen derivative 2d)
Affinity DataIC50:  5.44E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197342(CHEMBL3912637)
Affinity DataIC50:  6.27E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197300(CHEMBL3912164 | ebselen derivative 2e)
Affinity DataIC50:  6.79E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197346(CHEMBL3919905)
Affinity DataIC50:  7.57E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197298(CHEMBL3947694)
Affinity DataIC50:  8.85E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197343(CHEMBL3940582)
Affinity DataIC50:  9.13E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197349(CHEMBL3983492 | ebselen derivative 1e)
Affinity DataIC50:  9.98E+3nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197301(CHEMBL3922662 | ebselen derivative 1d)
Affinity DataIC50:  1.02E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM106945(US8592468, EbSe3)
Affinity DataIC50:  1.04E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197350(CHEMBL3964347)
Affinity DataIC50:  1.09E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197351(CHEMBL3894620)
Affinity DataIC50:  1.39E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197296(CHEMBL3894673)
Affinity DataIC50:  2.43E+4nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMicrotubule-associated protein 2(Human)
Wroclaw University of Technology

Curated by ChEMBL
LigandPNGBDBM50197345(CHEMBL3931557)
Affinity DataIC50:  1.19E+5nMAssay Description:Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed