TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.60nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 2.40nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 2.80nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 5.70nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 5.80nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 29nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 62nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 64nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 118nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 206nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 252nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 328nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 332nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 404nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 440nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 628nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 633nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.08E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.11E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 1.95E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 2.72E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 3.46E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis S.r.l.
Curated by ChEMBL
Promidis S.r.l.
Curated by ChEMBL
Affinity DataIC50: 5.23E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Istituto di Scienze e Tecnologie Molecolari (ISTM)
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged XIAP BIR3 domain (241 to 356 residues) expressed in Escherichia coli BL21(DE3) cells afte...More data for this Ligand-Target Pair
