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TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284924(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284924(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 15nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM686([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,10-Dimethyleth...)
Affinity DataIC50: 30nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM679(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 40nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284937({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-4...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM680((phenylmethyl)propyl]carbamic Acid, 1,1-Dimethylet...)
Affinity DataIC50: 40nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284925({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284937({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-4...)
Affinity DataIC50: 40nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM676(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 49nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM671([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 50nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM691(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 50nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284929({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 50nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM681([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 60nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM672(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 60nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284930({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284930({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 60nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM674([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 64nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM675([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 72nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM693(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 80nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM683(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 85nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM692(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 86nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM685([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 90nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM670(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 90nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM684(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 100nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM918(BMS-186318 analog 4 | tert-butyl N-[(2S,3R)-4-{[(2...)
Affinity DataIC50: 100nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM918(BMS-186318 analog 4 | tert-butyl N-[(2S,3R)-4-{[(2...)
Affinity DataIC50: 100nMpH: 5.5 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM682(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 100nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM673([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 110nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284932({(1S,2R)-1-Benzyl-3-[(2R,3S)-3-(2,4-dihydroxy-2,3,...)
Affinity DataIC50: 120nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM677(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 120nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM914(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 125nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM914(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 125nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284932({(1S,2R)-1-Benzyl-3-[(2R,3S)-3-(2,4-dihydroxy-2,3,...)
Affinity DataIC50: 130nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM666([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 130nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM688(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-4-[3-(benzyloxy)...)
Affinity DataIC50: 140nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM678([1S-[1R*,2S*(2S*,3R*)]]-[4-[4-(Carboxymethoxy)phen...)
Affinity DataIC50: 150nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM668([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 200nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284934(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284934(((1S,2R)-1-Benzyl-2-hydroxy-3-{(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 220nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284935({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 260nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM689(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-4-{4-[3-(1,3-ben...)
Affinity DataIC50: 280nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM687(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-4-[4-(benzyloxy)...)
Affinity DataIC50: 300nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM669([1S-[1R*,2S*(2S*,3R*)]]-[3-[[3-[[(1,1-Dimethyletho...)
Affinity DataIC50: 300nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM690(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-4-[4-(1,3-benzox...)
Affinity DataIC50: 320nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284931({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 320nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM665(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 400nMpH: 5.5 T: 2°CAssay Description:IC50 values are determined by inhibition of the cleavage of the peptidic substrate [V-S-Q-N-(beta-naphthylalanine)-P-I-V]. The IC50 value represents ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM923(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-[(tert-butylca...)
Affinity DataIC50: 400nMpH: 5.5 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50284926({(1S,2R)-1-Benzyl-2-hydroxy-3-[(2R,3S)-2-hydroxy-3...)
Affinity DataIC50: 450nMAssay Description:In vitro inhibition of HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails Article

TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM917(tert-butyl N-[(2S,3R)-4-{[(2R,3S)-3-{[(tert-butoxy...)
Affinity DataIC50: 500nMpH: 5.5 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Bristol-Myers Squibb

LigandPNGBDBM922((1S-(1R*,2S*(2S*,3R*)))-[3-[[3-[[[(1,1-Dimethyleth...)
Affinity DataIC50: 700nMpH: 5.5 T: 2°CAssay Description:Sensitivity of HIV-1 protease activity to protease inhibitors was determined by a peptide substrate cleavage assay. Protease products were analyzed o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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