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TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  0.0400nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB


TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36810(BMS753 | US9963439, BMS753)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  1nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor alpha [200-419]/gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36811(BMS614)
Affinity DataKi:  1nM ΔG°:  -47.8kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor gamma [183-417](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM31889(BMS 961 | BMS270394 | BMS961)
Affinity DataKi:  1.5nM ΔG°:  -46.8kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36810(BMS753 | US9963439, BMS753)
Affinity DataKi:  2nM ΔG°:  -46.2kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha [200-419](Human)
Institute of Genetics and Molecular and Cellular Biology (Igbmc)

LigandPNGBDBM36811(BMS614)
Affinity DataKi:  2.5nM ΔG°:  -45.6kJ/molepH: 8.0 T: 4°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB


TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  3.30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  3.80nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  4.10nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedMMDB


TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  5.90nMAssay Description:Selective activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  6.5nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  8.30nMAssay Description:Selective activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  11nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)
Affinity DataKi:  12nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  16nMAssay Description:Selective activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061625(4-[(5,5,8,8-tetramethyl-5,6,7,8-tetrahydronaphthal...)
Affinity DataKi:  30nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  50nMAssay Description:Selective activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  54nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  120nMAssay Description:Agonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  130nMAssay Description:Selective activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKi:  180nMAssay Description:Selective activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061616(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  220nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  320nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)
Affinity DataKi:  330nMAssay Description:Agonisticactivity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  400nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  490nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  500nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  620nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  640nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  680nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  790nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  810nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  900nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061618(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-thi...)
Affinity DataKi:  900nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  980nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.00E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.00E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  1.20E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.30E+3nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061616(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.40E+3nMAssay Description:Antagonistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.50E+3nMAssay Description:Antagonistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.60E+3nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-beta(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061615(4-(10,10,13,13,15-Pentamethyl-11,12,13,15-tetrahyd...)
Affinity DataKi:  1.70E+3nMAssay Description:Antagonistic activity of the compound towards retinoid X receptor-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061619(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5H-13...)
Affinity DataKi:  1.80E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061624(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  1.90E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061621(4-(5,7,7,10,10-Pentamethyl-7,8,9,10-tetrahydro-5H-...)
Affinity DataKi:  2.00E+3nMAssay Description:Synergistic activity of the compound towards retinoic acid receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-gamma(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  2.10E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetRetinoic acid receptor RXR-alpha(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50061617(4-(7,7,10,10-Tetramethyl-7,8,9,10-tetrahydro-5-oxa...)
Affinity DataKi:  3.80E+3nMAssay Description:Synergistic activity of the compound towards retinoid X receptor-alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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