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TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM86192(CAS_197801-88-0 | CHEMBL2165203 | SN003)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to CRFR1 by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50152162(CHEMBL188844 | CHEMBL2165204 | [3-(6-Dimethylamino...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to CRFR1 by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50395823(CHEMBL2165205)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to CRFR1 by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50395822(CHEMBL1762817)
Affinity DataKi:  2nMAssay Description:Binding affinity to CRF1 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50395822(CHEMBL1762817)
Affinity DataKi:  2nMAssay Description:Binding affinity to CRFR1 by autoradiographyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177574(3-(4-(2-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177568(3-(4-(benzyloxy)phenylsulfonyl)-N-mesityl-6-methyl...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177576(3-(4-(3,5-dimethoxybenzyloxy)phenylsulfonyl)-N-mes...)
Affinity DataKi:  34nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177581(CHEMBL437893 | methyl 3-((4-(2-(mesitylamino)-6-me...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177584(3-(4-ethylphenylsulfonyl)-N-mesityl-6-methylpyridi...)
Affinity DataKi:  52nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177572(3-(4-(3-methoxybenzyloxy)phenylsulfonyl)-N-mesityl...)
Affinity DataKi:  58nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177582(3-((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfon...)
Affinity DataKi:  75nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177570(3-(4-(allyloxy)phenylsulfonyl)-N-mesityl-6-methylp...)
Affinity DataKi:  119nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218669(CHEMBL97868)
Affinity DataKi:  127nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177588(3-(3-(benzyloxy)phenylsulfonyl)-N-mesityl-6-methyl...)
Affinity DataKi:  132nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218662(CHEMBL100943)
Affinity DataKi:  143nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177587(CHEMBL204967 | N-mesityl-6-methyl-3-tosylpyridin-2...)
Affinity DataKi:  145nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177575(4-((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfon...)
Affinity DataKi:  157nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218754(CHEMBL101574)
Affinity DataKi:  173nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177577(CHEMBL203744 | N-mesityl-3-(4-methoxyphenylsulfony...)
Affinity DataKi:  198nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218684(CHEMBL99741)
Affinity DataKi:  223nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177571(CHEMBL201470 | N-mesityl-3-(3-methoxyphenylsulfony...)
Affinity DataKi:  249nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177586(CHEMBL382347 | N-mesityl-6-methyl-3-(4-(pyridin-2-...)
Affinity DataKi:  250nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177583(CHEMBL201966 | N-mesityl-6-methyl-3-(4-(trifluorom...)
Affinity DataKi:  268nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218683(CHEMBL98643)
Affinity DataKi:  324nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177589(5-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfony...)
Affinity DataKi:  395nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218680(CHEMBL318652)
Affinity DataKi:  485nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218753(CHEMBL101093)
Affinity DataKi:  492nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218687(CHEMBL327285)
Affinity DataKi:  597nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218685(CHEMBL316839)
Affinity DataKi:  623nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177573(4-(4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfony...)
Affinity DataKi:  635nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218661(CHEMBL98693)
Affinity DataKi:  671nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218681(CHEMBL98091)
Affinity DataKi:  825nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177567(3-(4-chlorobenzylsulfonyl)-N-mesityl-6-methylpyrid...)
Affinity DataKi:  857nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177579((4-(2-(mesitylamino)-6-methylpyridin-3-ylsulfonyl)...)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218679(CHEMBL100168)
Affinity DataKi:  1.14E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218759(CHEMBL99155)
Affinity DataKi:  1.36E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218975(CHEMBL431229)
Affinity DataKi:  1.54E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177566(CHEMBL203609 | N-mesityl-4,6-dimethyl-3-tosylpyrid...)
Affinity DataKi:  1.78E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218678(CHEMBL317436)
Affinity DataKi:  2.22E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218797(CHEMBL320384)
Affinity DataKi:  2.42E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218686(CHEMBL318729)
Affinity DataKi:  2.88E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1/2(Rat)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50218660(CHEMBL99550)
Affinity DataKi: >3.00E+3nMAssay Description:Binding affinity at corticotropin releasing hormone receptor in rat frontal cortex homogenates by [125I]Tyr-o-CRF displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177580(CHEMBL204014 | N-mesityl-4,6-dimethyl-3-(m-tolylsu...)
Affinity DataKi:  5.17E+3nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177585(CHEMBL371013 | N-mesityl-4,6-dimethyl-3-(o-tolylsu...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177578(CHEMBL382015 | N-mesityl-6-methyl-5-tosylpyridin-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCorticotropin-releasing factor receptor 1(Rat)
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50177569(CHEMBL381898 | N-mesityl-4,6-dimethyl-3-(phenylsul...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]Tyr-o-CRF from CRF1 receptor in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM610463(BDBM610464 | BDBM610465 | N-(4-(2-Methylmorpholino...)
Affinity DataIC50:  0.0900nMAssay Description:The kinase assay was performed in V-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme, subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails US Patent

TargetGlycogen synthase kinase-3 alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM610453(2-Phenyl-N-(4-(2,2,2-trifluoroethoxy)pyridin-3-yl)...)
Affinity DataIC50:  0.0900nMAssay Description:Inhibition of full length GST-tagged human recombinant GSK3-alpha using FL-KRREILSRRP[ps]ERYR-NH2 as substrate incubated for 20 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM50613245(CHEMBL5266553)
Affinity DataIC50:  0.100nMAssay Description:Inhibition of full length GST-tagged human recombinant GSK3-alpha using FL-KRREILSRRP[ps]ERYR-NH2 as substrate incubated for 20 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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