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TargetApelin(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50009575(CHEMBL3234446)
Affinity DataKi:  0.0400nMAssay Description:Displacement of [125I]-pE13F from human apelin receptor expressed in CHO cell membranes after 1 hr by gamma counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.0955nMAssay Description:Displacement of [3H]NMS from EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 22 hrs by liquid scinti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50241132(3-Hydroxy-2-phenyl-propionic acid 9-methyl-3-oxa-9...)
Affinity DataKi:  0.170nMAssay Description:Competitive inhibition of EGFP-fused human M1 receptor N-terminal truncated at 17 residues expressed in HEK293 cells after 4 hrs by FRET assay in pre...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.210nMAssay Description:Competitive binding to human oxytocin receptor by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459408(CHEMBL3307200)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.450nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  0.480nMAssay Description:Displacement of [3H]AVP from V1A receptor in Wistar rat liver membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1b receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1b receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]-AVP from human V2 receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  0.570nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  0.589nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  0.603nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor entirely in guinea pig ileumMore data for this Ligand-Target Pair
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077141(CHEMBL3416758)
Affinity DataKi:  0.670nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1a receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Competitive binding to oxytocin receptor (unknown origin) by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  0.790nMAssay Description:Binding affinity to OTR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397209(CHEMBL2172291)
Affinity DataKi:  0.830nMAssay Description:Displacement of [3H]-AVP from SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  1nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.36nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 mins by saturation binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50014407(2-(piperazin-1-yl)quinoline | 2-Piperazin-1-yl-qui...)
Affinity DataKi:  1.40nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptor in the rabbit heartMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.48nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM35667(AVP | CHEMBL373742 | US10131692, 44 (AVP) | [3H]Ar...)
Affinity DataKi:  1.65nMAssay Description:Displacement of [3H]-AVP from human oxytocin receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397210(CHEMBL2172290)
Affinity DataKi:  1.93nMAssay Description:Displacement of [3H]-AVP from SNAP-tagged vasopressin V2 receptor expressed in HEK293 cells by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50459401(CHEMBL4210854)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  2.68nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]-AVP from human V1A receptor expressed in CHO cell membranes by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]-AVP from human vasopressin V1a receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  2.74nMAssay Description:Displacement of [3H]AVP from human vasopressin V1a receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM85095(CAS_151171 | CONIVAPTAN | NSC_151171 | YM087)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]AVP from V2 receptor in Wistar rat kidney membranes incubated for 60 mins by microplate scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  3.20nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.31nMAssay Description:Potency at neuronal 5-hydroxytryptamine 3 receptors in the rabbit heartMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397215(CHEMBL2172295)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397206(CHEMBL2172289)
Affinity DataKi:  5.69nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  6.20nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50307120(5-[4-[(1,1'-Biphenyl-2-ylcarbonyl)amino]-3-methylb...)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]AVP from human vasopressin V2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50077140(CHEMBL3416757)
Affinity DataKi:  6.60nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  6.60nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  7.20nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50307117(CHEMBL603708 | N-(4-(2,3,4,5-tetrahydro-1H-benzo[b...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397213(CHEMBL2172391)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Umr7200 Cnrs/Universit£

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397219(CHEMBL2172285)
Affinity DataKi:  8.80nMAssay Description:Binding affinity to human muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50151212(CHEMBL2368393 | difluoro(2-{[(2Z)-1-methyl-5-[2-({...)
Affinity DataKi:  8.80nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50151218(CHEMBL2368392 | difluoro(2-{[(2Z)-1-methyl-5-(2-{[...)
Affinity DataKi:  8.90nMAssay Description:Inhibition of [3H]QNB binding to human muscarinic receptor M1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50397210(CHEMBL2172290)
Affinity DataKi:  9.02nMAssay Description:Displacement of [3H]-AVP from human vasopressin V2 receptor expressed in CHO cells after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A/3B(Rat)
Merrell Dow Research Institute

Curated by ChEMBL
LigandPNGBDBM50000483((BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid ...)
Affinity DataKi:  9.10nMAssay Description:Binding affinity to 5-hydroxytryptamine 3 receptor of neuronal in the afferent rabbit vagusMore data for this Ligand-Target Pair
TargetOxytocin receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM50205990(CHEMBL395429 | OXYTOCIN)
Affinity DataKi:  9.5nMAssay Description:Competitive binding to SNAP-tagged oxytocin receptor (unknown origin) expressed in HEK293 cells incubated for 1 hr at RT followed by 4 hrs at 4 degC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
University of Strasburg

Curated by ChEMBL
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.70nMAssay Description:Binding affinity to vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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