Compile Data Set for Download or QSAR
Found 470 with Last Name = 'hipskind' and Initial = 'pa'
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075807(1-(3-{1-[2-(4-Iodo-phenyl)-ethyl]-piperidin-4-yl}-...)
Affinity DataKi:  0.0520nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075796(2-Phenoxymethyl-4-(3-piperidin-1-yl-propoxy)-1-{3-...)
Affinity DataKi:  0.106nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075811(3-(4-{3-[2-Phenoxymethyl-4-(3-piperidin-1-yl-propo...)
Affinity DataKi:  0.112nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075803(4-(4-{3-[2-Phenoxymethyl-4-(3-piperidin-1-yl-propo...)
Affinity DataKi:  0.132nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186291(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-...)
Affinity DataKi:  0.170nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075812(2-Phenoxymethyl-1-{3-[1-((Z)-3-phenyl-allyl)-piper...)
Affinity DataKi:  0.183nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075809(1-[3-(1-Phenethyl-piperidin-4-yl)-propyl]-2-phenox...)
Affinity DataKi:  0.191nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186270(2-benzyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tet...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186278(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186290(3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075797(1-{3-[1-(2-Cyclohexyl-ethyl)-piperidin-4-yl]-propy...)
Affinity DataKi:  0.285nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075806(1-{3-[1-(3-Methyl-butyl)-piperidin-4-yl]-propyl}-2...)
Affinity DataKi:  0.290nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075802(4-[2-(4-{3-[2-Phenoxymethyl-4-(3-piperidin-1-yl-pr...)
Affinity DataKi:  0.313nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186309(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186269(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186292(2-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075799(2-Phenoxymethyl-1-{3-[1-(3-phenyl-propyl)-piperidi...)
Affinity DataKi:  0.361nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075798(1-[3-(1-Cyclohexylmethyl-piperidin-4-yl)-propyl]-2...)
Affinity DataKi:  0.393nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186292(2-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.460nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186316(2-(phenylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-1...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186306(3-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186283(2-ethyl-6-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186309(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186293(7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetrahydrois...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186269(2-ethyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-tetr...)
Affinity DataKi:  0.640nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075795(1-[3-(1-But-3-enyl-piperidin-4-yl)-propyl]-2-pheno...)
Affinity DataKi:  0.707nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186311(3-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  0.720nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075808(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  0.75nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  0.75nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  0.75nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186270(2-benzyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tet...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075804(1-[3-(1-Isobutyl-piperidin-4-yl)-propyl]-2-phenoxy...)
Affinity DataKi:  0.829nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186291(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-1,2,3,4-...)
Affinity DataKi:  0.890nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186306(3-(cyclohexylmethyl)-7-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  0.970nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186296(2-(cyclohexylmethyl)-6-(3-(piperidin-1-yl)propoxy)...)
Affinity DataKi:  1.01nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186290(3-ethyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-tetr...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186278(2-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  1.29nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50060726(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075801(1-[3-(1-Methyl-piperidin-4-yl)-propyl]-2-phenoxyme...)
Affinity DataKi:  1.60nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186311(3-isopropyl-7-(3-(piperidin-1-yl)propoxy)-2,3,4,5-...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075800(1-[3-(1-Allyl-piperidin-4-yl)-propyl]-2-phenoxymet...)
Affinity DataKi:  1.60nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075810(1-[3-(1-Isopropyl-piperidin-4-yl)-propyl]-2-phenox...)
Affinity DataKi:  1.60nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50065468(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-pro...)
Affinity DataKi:  1.70nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50065468(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-pro...)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity towards human neuropeptide Y receptor type 1, determined by measuring its ability to displace [125]peptide YYMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50060725(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  1.80nMAssay Description:Ability of the compound to reverse Neuropeptide Y receptor type 1-induced inhibition of forskolin-induced inhibition of forskolin-stimulated cAMPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50060724(2-[1,4']Bipiperidinyl-1'-yl-1-[2-(4-chloro-phenoxy...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity for Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50065468(2-(4-Chloro-phenoxymethyl)-4-(3-piperidin-1-yl-pro...)
Affinity DataKi:  2nMAssay Description:Binding affinity of the compound at cloned Neuropeptide Y receptor type 1 expressed in AV-12 cells is evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186281((6-(3-(piperidin-1-yl)propoxy)-3,4-dihydroisoquino...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50186295(2-(methylsulfonyl)-7-(3-(piperidin-1-yl)propoxy)-2...)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human cloned H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 1(Homo sapiens (Human))
Eli Lilly and Company

Curated by ChEMBL
LigandPNGBDBM50075805(2-Phenoxymethyl-4-(3-piperidin-1-yl-propoxy)-1-(3-...)
Affinity DataKi:  4.5nMAssay Description:Ability to displace [125I]-peptide YY binding to cloned human Neuropeptide Y receptor type 1 expressed in AV-12 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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