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TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185909(2-(3-((1-(3-(2-chlorophenoxy)benzyl)piperidin-4-yl...)
Affinity DataIC50: 1nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185912(2-(4-{1-[3-(2-chloro-phenoxy)-benzyl]-piperidin-4-...)
Affinity DataIC50: 4nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185905(4-phenyl-piperidine-4-carboxylic acid {1-[3-(2-met...)
Affinity DataIC50: 11nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185904((+/-) 3-phenyl-pyrrolidine-3-carboxylic acid {1-[3...)
Affinity DataIC50: 22nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138590(2-(7-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138578(2-(7-Hydroxy-1-methyl-3,4-dihydro-1H-isoquinolin-2...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138594(2-(5-Hydroxy-1,3-dihydro-isoindol-2-ylmethyl)-N-(4...)
Affinity DataIC50: 33nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138558(2-[(6-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-ylam...)
Affinity DataIC50: 43nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185910(1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[...)
Affinity DataIC50: 43nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185907(N-{1-[3-(2-methoxy-phenoxy)-benzyl]-piperidin-4-yl...)
Affinity DataIC50: 55nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138584(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-((E...)
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetC-C chemokine receptor type 8(Human)
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50185908(1-ethyl-4-phenyl-piperidine-4-carboxylic acid {1-[...)
Affinity DataIC50: 56nMAssay Description:Inhibition of I309-induced chemotaxis in L1.2 cells expressing CCR8More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138559(2-(7-Hydroxy-1,2,4,5-tetrahydro-benzo[d]azepin-3-y...)
Affinity DataIC50: 58nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138556(2-(7-Hydroxy-3-methyl-3,4-dihydro-1H-isoquinolin-2...)
Affinity DataIC50: 67nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138565(N-[4-(4-Chloro-phenyl)-butyl]-2-{[2-(4-hydroxy-phe...)
Affinity DataIC50: 77nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138555(2-[(6-Hydroxy-1,2,3,4-tetrahydro-naphthalen-2-ylam...)
Affinity DataIC50: 81nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138561(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 86nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138569(2-(7-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 89nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138572(N-[4-(3-Chloro-phenyl)-butyl]-2-{[2-(4-hydroxy-phe...)
Affinity DataIC50: 99nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138587(N-[4-(3,4-Dichloro-phenyl)-butyl]-2-{[2-(4-hydroxy...)
Affinity DataIC50: 120nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138592(2-(6-Hydroxy-3,4-dihydro-1H-isoquinolin-2-ylmethyl...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138576(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-[4-...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138575(2-[(2-Hydroxy-6,7,8,9-tetrahydro-5H-benzocyclohept...)
Affinity DataIC50: 130nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138564(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138562(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-[4-...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138596(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 170nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138586(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-((Z...)
Affinity DataIC50: 300nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138579(2-(7-Hydroxy-1,3,4,5-tetrahydro-benzo[c]azepin-2-y...)
Affinity DataIC50: 320nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138566(2-{[2-(3-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 330nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138554(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-[4-...)
Affinity DataIC50: 370nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155833(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 370nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 400nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155832(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 440nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155822(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 500nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155821(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 610nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138577(2-{[3-(4-Hydroxy-phenyl)-propylamino]-methyl}-N-(4...)
Affinity DataIC50: 670nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155825(3-[4-(2,4-Bis-trifluoromethyl-benzyloxy)-3-methoxy...)
Affinity DataIC50: 750nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155820(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(5...)
Affinity DataIC50: 800nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155820(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(5...)
Affinity DataIC50: 800nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155830(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(4...)
Affinity DataIC50: 920nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155830(2-Cyano-N-(5-ethyl-[1,3,4]thiadiazol-2-yl)-3-[4-(4...)
Affinity DataIC50: 920nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138589(2-[(4-Hydroxy-benzylamino)-methyl]-N-(4-phenyl-but...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138567(2-{[2-(4-Methoxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138585(2-{[2-(2-Hydroxy-phenyl)-ethylamino]-methyl}-N-(4-...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50404282(CHEMBL2112891)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155815(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155828(6-[1-{4-[2-(2,6-Dimethyl-phenoxy)-ethoxy]-3-methox...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of estrogen-related receptor alpha in FP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSteroid hormone receptor ERR1(Human)
X-Ceptor Therapeutics

Curated by ChEMBL
LigandPNGBDBM50155817(2-Cyano-3-{4-[2-(2,6-dimethyl-phenoxy)-ethoxy]-3-m...)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of estrogen-related receptor alpha Gal4 activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50138591(2-{[2-(4-Hydroxy-phenyl)-ethylamino]-methyl}-N-(3-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against human glycine transporter type 2 (hGlyT2) expressed in Chinese hamster ovary (CHO) cell lineMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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