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TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101825((Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101823(4-(2-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-...)
Affinity DataKi: >0.000100nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101827((Z)-7-{(1R,2R,3R)-2-[(E)-(S)-4-(1-Ethyl-cyclobutyl...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101826((Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101823(4-(2-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1-...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101833((Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101832((E)-7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1...)
Affinity DataKi: >0.000100nMAssay Description:Binding affinity towards mouse Prostanoid EP3 receptor in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101832((E)-7-{(1R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4-(1...)
Affinity DataKi: >0.000100nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProstacyclin receptor(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50101825((Z)-7-{(1R,2R,3R)-3-Hydroxy-2-[(E)-(S)-4-hydroxy-4...)
Affinity DataKi: >0.000100nMAssay Description:Effective concentration which increases intracellular c-AMP production in human Prostanoid IP receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578123(CHEMBL4872591)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578124(CHEMBL4866325)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578111(CHEMBL4861425)
Affinity DataEC50:  0.0130nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578122(CHEMBL4849848)
Affinity DataEC50:  0.0140nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578121(CHEMBL4860633)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578128(CHEMBL4873269)
Affinity DataEC50:  0.0170nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578126(CHEMBL4853282)
Affinity DataEC50:  0.0190nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578120(CHEMBL4858892)
Affinity DataEC50:  0.0270nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50272772(CHEMBL1680 | 10-(4-Amino-butyl)-19-(2-amino-3-phen...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578109(CHEMBL4863880)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578110(CHEMBL4845867)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578118(CHEMBL4870834)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578129(CHEMBL4862195)
Affinity DataEC50:  0.0480nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50223276(CHEMBL65426)
Affinity DataIC50: 0.0510nMAssay Description:Inhibition of phosphodiesterase 4 (PDE4) prepared from human U937 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataKi:  0.0680nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286892(1-[(R)-1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pheny...)
Affinity DataIC50: 0.0700nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578127(CHEMBL4876263)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578119(CHEMBL4851978)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50223272(CHEMBL67668)
Affinity DataIC50: 0.0800nMAssay Description:Inhibition of phosphodiesterase 4 (PDE4) prepared from human U937 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578125(CHEMBL4878917)
Affinity DataEC50:  0.0810nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataKi:  0.0970nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286884(1-{1-[2-(1-Methyl-cyclopentyl)-2-oxo-ethyl]-2-oxo-...)
Affinity DataIC50: 0.100nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056102(YF-476 | 1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo...)
Affinity DataIC50: 0.100nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578117(CHEMBL4854548)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Ability to displace [125I]CCK-8 from gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056103(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056099(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-pyridi...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056093(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataIC50: 0.110nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056101(CHEMBL115121 | YM022 Racemate | YM022 | 1-[(R)-2-O...)
Affinity DataKi:  0.110nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2011
Entry Details
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578116(CHEMBL4862497)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286903(1-[1-(2-Cyclopentyl-2-oxo-ethyl)-2-oxo-5-pyridin-2...)
Affinity DataIC50: 0.120nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50286897(1-[2-Oxo-1-(2-oxo-2-o-tolyl-ethyl)-5-pyridin-2-yl-...)
Affinity DataIC50: 0.130nMAssay Description:Binding affinity towards gastrin/Cholecystokinin type B receptor from rat brain using [125I]CCK-8 as the radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578114(CHEMBL4862717)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056092(1-(3-Diethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-2...)
Affinity DataIC50: 0.140nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056091(1-[1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl-2,3...)
Affinity DataIC50: 0.160nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056089(1-[(R)-1-(3,3-Dimethyl-2-oxo-butyl)-2-oxo-5-phenyl...)
Affinity DataIC50: 0.170nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4A/4B/4C/4D(Human)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50223263(CHEMBL291889)
Affinity DataIC50: 0.180nMAssay Description:Inhibition of phosphodiesterase 4 (PDE4) prepared from human U937 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/22/2018
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Yamanouchi Pharmaceutical

Curated by PDSP Ki Database
LigandPNGBDBM50056095(1-(3-Dimethylamino-phenyl)-3-[(R)-1-(3,3-dimethyl-...)
Affinity DataIC50: 0.200nMAssay Description:Inhibitory concentration against radioligand [125I]CCK-8 binding to gastrin/Cholecystokinin type B receptor from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 2(Human)
Ono Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50578113(CHEMBL4854239)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at human SSTR2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation measured after 30 mins by Glo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
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