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TargetAcetylcholinesterase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284042(2-(1-{2-[(5-Piperidin-1-ylmethyl-furan-2-ylmethyl)...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against acetylcholinesterase (AChE) from rat brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article

Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50032282(4-(2-{(E)-3-[1-(1-Propyl-butyl)-1H-indol-5-yl]-but...)
Affinity DataIC50: 2.30nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50010960((E)-7-Phenyl-7-pyridin-3-yl-hept-6-enoic acid | CV...)
Affinity DataIC50: 2.90nMAssay Description:Activity against TXA2 synthase in bovine platelet microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50032297(4-[2-((E)-3-{1-[Bis-(4-fluoro-phenyl)-methyl]-1H-i...)
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470304(CHEMBL98478)
Affinity DataIC50: 3.60nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50047486(11-(Pyridin-3-ylmethylsulfanyl)-6,11-dihydro-diben...)
Affinity DataIC50: 4nMAssay Description:Activity against TXA2 synthase in bovine platelet microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50032281(4-(2-{(E)-3-[1-(1-Propyl-pentyl)-1H-indol-5-yl]-bu...)
Affinity DataIC50: 4.10nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50047491(Sodium; (E)-2-methyl-3-(4-pyridin-3-ylmethyl-pheny...)
Affinity DataIC50: 4.30nMAssay Description:Activity against TXA2 synthase in bovine platelet microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50032288(4-{2-[(E)-3-(1-Benzhydryl-1H-indol-5-yl)-but-2-eno...)
Affinity DataIC50: 5.60nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056538({3-[(5-CHLORO-1,3-BENZOTHIAZOL-2-YL)METHYL]-2,4-DI...)
Affinity DataIC50: 5.70nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470291(CHEMBL95410)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470283(CHEMBL421752)
Affinity DataIC50: 6.30nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470301(CHEMBL99824)
Affinity DataIC50: 7.10nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470289(CHEMBL96030)
Affinity DataIC50: 7.20nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470272(CHEMBL431270)
Affinity DataIC50: 7.80nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50032264(4-(2-{(E)-3-[1-(1-Isobutyl-3-methyl-butyl)-1H-indo...)
Affinity DataIC50: 8nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470263(CHEMBL99811)
Affinity DataIC50: 8.10nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470268(CHEMBL319506)
Affinity DataIC50: 8.80nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470293(CHEMBL329690)
Affinity DataIC50: 8.80nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470260(CHEMBL99860)
Affinity DataIC50: 9.10nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470274(CHEMBL319549)
Affinity DataIC50: 9.30nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470277(CHEMBL97506)
Affinity DataIC50: 9.80nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470303(CHEMBL319505)
Affinity DataIC50: 9.80nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056534([3-(4-Chloro-benzothiazol-2-ylmethyl)-2,4-dioxo-3,...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056531([3-(4-Chloro-benzothiazol-2-ylmethyl)-2,4,5-trioxo...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284039(2-(1-{2-[(5-Piperidin-1-ylmethyl-furan-2-ylmethyl)...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against acetylcholinesterase (AChE) from rat brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article

Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470299(CHEMBL95946)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470302(CHEMBL29925)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50047487(11-(2-Pyridin-3-yl-ethylidene)-6,11-dihydro-dibenz...)
Affinity DataIC50: 14nMAssay Description:Activity against TXA2 synthase in bovine platelet microsomeMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284041(2-(1-(3-Methoxy-phenyl)-3-{2-[(5-piperidin-1-ylmet...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against acetylcholinesterase (AChE) from rat brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article

TargetAcetylcholinesterase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284043(2-(1-Phenyl-3-{2-[(5-piperidin-1-ylmethyl-furan-2-...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against acetylcholinesterase (AChE) from rat brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article

Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470267(CHEMBL316858)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056540([3-(5-Chloro-benzothiazol-2-ylmethyl)-2,4,5-trioxo...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056535([3-(4-Chloro-3-nitro-benzyl)-2,4,5-trioxo-imidazol...)
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470264(CHEMBL443496)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470266(CHEMBL100314)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470292(CHEMBL100318)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284040(2-(1-(4-Methoxy-phenyl)-3-{2-[(5-piperidin-1-ylmet...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against acetylcholinesterase (AChE) from rat brain was determinedMore data for this Ligand-Target Pair
In DepthDetails Article

Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470271(CHEMBL327722)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50049730(Epalrestat | 2-(5-(2-methyl-3-phenylallylidene)-4-...)
Affinity DataIC50: 21nMAssay Description:In vitro inhibitory activity against partially purified rat lens Aldose reductase at a dose of 5e-7MMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50049730(Epalrestat | 2-(5-(2-methyl-3-phenylallylidene)-4-...)
Affinity DataIC50: 21nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50022775(m-Trimethylammoniumphenyldimethylcarbamate | Prost...)
Affinity DataIC50: 22nMAssay Description:Inhibition of guinea pig acetylcholinesteraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470284(CHEMBL99473)
Affinity DataIC50: 23nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056533([3-(4-Chloro-3-nitro-benzyl)-2,4-dioxo-imidazolidi...)
Affinity DataIC50: 24nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470262(CHEMBL431435)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470279(CHEMBL327521)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470285(CHEMBL99300)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
Target3-oxo-5-alpha-steroid 4-dehydrogenase 1/2(Rat)
Kyowa Hakko Kogyo

Curated by ChEMBL
LigandPNGBDBM50470290(CHEMBL328182)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against Steroid 5-alpha-reductase in prostates from male ratsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056527([3-(4-Chloro-3-nitro-benzyl)-2,4-dioxo-3,4-dihydro...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetAldo-keto reductase family 1 member B1(Rat)
Nippon Zoki Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50056532([3-(3-Nitro-benzyl)-4,5-dioxo-2-thioxo-imidazolidi...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against rat lens aldose reductase(AR).More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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