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TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064089(4-hydroxymethyl-7,10-diisopropyl-8,10,13-trimethyl...)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  0.430nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081077(CHEMBL216658 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081078(CHEMBL374446 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50081076(CHEMBL414278 | Dicarba-Closo-Dodecaborane analogue)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064090((S)-2-Decyl-5-hydroxymethyl-1-methyl-1,4,5,6-tetra...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064091((2S,5S)-9-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.42nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073876((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-met...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064092(5'-hydroxymethyl-2'-isopropyl-1',4,4-trimethyl-(2'...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073875((1S,4S,5aS,9aS)-1,7,7-Tributyl-4-hydroxymethyl-5a-...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064094(5'-hydroxymethyl-2'-isopropyl-1'-methyl-(2'S,5'S)-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073873((1S,4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-1,5a-d...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V1a receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  32nMAssay Description:Binding affinity of the compound towards Vasopressin V1a receptor in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064093((7S,10S)-10-Hydroxymethyl-7-isopropyl-4,4,6-trimet...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073874((4S,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073878((4R,5aS,9aS)-7,7-Dibutyl-4-hydroxymethyl-5a-methyl...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073872((4S,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073870((4R,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073877((4S,5aS,5bS,7aR,8R,10aS,10bR,12aS)-8-(1,5-Dimethyl...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C alpha type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50073871((4R,5aS,5bS,7aS,10aS,10bS,12aS)-4-Hydroxymethyl-5a...)
Affinity DataKi: >500nMAssay Description:Displacement of [3H]-PDBu from human recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50057513((2S,5S)-5-Hydroxymethyl-2-isopropyl-1-methyl-1,4,5...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064088((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,6-trimet...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetProtein kinase C delta type(Human)
University of Tokyo

Curated by ChEMBL
LigandPNGBDBM50064095((7S,10S)-10-Hydroxymethyl-7-isopropyl-1,1,4,4,6-pe...)
Affinity DataKi:  5.10E+3nMAssay Description:Displacement of [3H]-PDBu from recombinant Protein kinase C deltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V1a receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  1.40E+4nMAssay Description:Binding affinity of the compound towards Vasopressin V1a receptor in human liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094076(CHEMBL434654 | N-[4-(7-Chloro-2,3,4,5-tetrahydro-b...)
Affinity DataIC50:  0.950nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094079((4-Amino-2-methyl-phenyl)-(7-chloro-2,3,4,5-tetrah...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094068((2-Chloro-4-ethylamino-phenyl)-(7-chloro-2,3,4,5-t...)
Affinity DataIC50:  5nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094086((4-Allylamino-2-chloro-phenyl)-(2,3,4,5-tetrahydro...)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094082((2-Chloro-4-pyrrol-1-yl-phenyl)-(2,3,4,5-tetrahydr...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094066((2-Chloro-4-pyrazol-1-yl-phenyl)-(2,3,4,5-tetrahyd...)
Affinity DataIC50:  8.80nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094075((2-Chloro-4-pyrrolidin-1-yl-phenyl)-(2,3,4,5-tetra...)
Affinity DataIC50:  9nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094074((2-Chloro-4-dimethylamino-phenyl)-(7-chloro-2,3,4,...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094070(CHEMBL136109 | [2-Chloro-4-(3-methyl-pyrazol-1-yl)...)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094072((2-Chloro-4-pyrrolidin-1-yl-phenyl)-(7-chloro-2,3,...)
Affinity DataIC50:  16nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094089((2-Chloro-4-propylamino-phenyl)-(2,3,4,5-tetrahydr...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094067((2-Chloro-4-dimethylamino-phenyl)-(2,3,4,5-tetrahy...)
Affinity DataIC50:  18nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094077((2-Chloro-4-diethylamino-phenyl)-(2,3,4,5-tetrahyd...)
Affinity DataIC50:  19nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094078((4-Butylamino-2-chloro-phenyl)-(2,3,4,5-tetrahydro...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094087((2-Chloro-4-pentylamino-phenyl)-(2,3,4,5-tetrahydr...)
Affinity DataIC50:  31nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094069((2-Chloro-4-ethylamino-phenyl)-(2,3,4,5-tetrahydro...)
Affinity DataIC50:  34nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094083((2-Chloro-4-methylamino-phenyl)-(2,3,4,5-tetrahydr...)
Affinity DataIC50:  35nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094076(CHEMBL434654 | N-[4-(7-Chloro-2,3,4,5-tetrahydro-b...)
Affinity DataIC50:  38nMAssay Description:Binding affinity of the compound towards rat Vasopressin V2 receptor after peroral administration of the compoundMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094088(CHEMBL136790 | [2-Chloro-4-(3-methyl-pyrrolidin-1-...)
Affinity DataIC50:  51nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094073((2-Chloro-4-piperidin-1-yl-phenyl)-(2,3,4,5-tetrah...)
Affinity DataIC50:  120nMAssay Description:Inhibition of [3H]-AVP binding to human Vasopressin V2 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50094075((2-Chloro-4-pyrrolidin-1-yl-phenyl)-(2,3,4,5-tetra...)
Affinity DataIC50:  150nMAssay Description:Binding affinity of the compound towards rat Vasopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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