Report error Found 185 with Last Name = 'jadav' and Initial = 'ss'
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKd: >1.00E+5nMAssay Description:Binding affinity to HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKd: 1.70E+3nMAssay Description:Binding affinity to HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataKd: 720nMAssay Description:Binding affinity to HCV NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of DHCR7 (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Inhibition of HCV NS3/4a protease using Ac-DE-Dap(QXL520)-EE-Abu-shi-[COO]AS-C(5-FAMsp)-NH2 as substrate after 15 minsMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of HCV NS3/4a protease using Ac-DE-Dap(QXL520)-EE-Abu-shi-[COO]AS-C(5-FAMsp)-NH2 as substrate after 15 minsMore data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of HCV NS3/4a protease using Ac-DE-Dap(QXL520)-EE-Abu-shi-[COO]AS-C(5-FAMsp)-NH2 as substrate after 15 minsMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Inhibition of TNKS2 (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 4.30nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of HCV NS5B polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Inhibition of human DNA polymerase beta by fluorescence anisotropyMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Inhibition of HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 7.20nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of HCV NS5B polymeraseMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 9.40nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of CDK4/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of TNKS1 (unknown origin)More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CDK4 (S4 to E303 residues)/Cyclin D1 (Q4 to I295 residues) expressed in sf9 cells using RBCTF a...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D1(Human)
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of CDK6/cyclin D1 (unknown origin) using RBER-CHKtide as substrate measured after 1 hr by ADP-glo luminescence assayMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Binding affinity to HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Inhibition of TNKS2 (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of DHCR7 (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Inhibition of HCV NS3/4a proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 36nMAssay Description:The COX activity was assayed colorimetrically by monitoring the appearance of oxidized N,N,N',N'-tetramethyl-pphenylenediamine (TMPD) at 590 ...More data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 39nMAssay Description:Inhibition of HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of TNKS1 (unknown origin)More data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetGenome polyprotein/Non-structural protein 4A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Inhibition of HCV NS3/4a proteaseMore data for this Ligand-Target Pair
TargetRNA-directed RNA polymerase(Hepatitis C virus genotype 1b (isolate Con1) (HCV))
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 53nMAssay Description:Inhibition of HCV NS5B polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 58nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 97nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 160nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 188nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Human)
Gitam (Deemed To Be University)
Curated by ChEMBL
Gitam (Deemed To Be University)
Curated by ChEMBL
Affinity DataIC50: 303nMAssay Description:Inhibition of EBP (unknown origin)More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 340nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Human)
De Montfort University
Curated by ChEMBL
De Montfort University
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CDK4 (S4 to E303 residues)/Cyclin D1 (Q4 to I295 residues) expressed in sf9 cells using RBCTF a...More data for this Ligand-Target Pair
TargetNonstructural protein 5A(Hepacivirus C)
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Institute of Pharmaceutical Education and Research
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Binding affinity to HCV NS5A polymeraseMore data for this Ligand-Target Pair
