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TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086013(CHEMBL10009 | N-[2-(2-Methoxy-6H-isoindolo[2,1-a]i...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50114716(CHEMBL329263 | N-[2-(2-Benzyl-5-methoxy-benzofuran...)
Affinity DataKi:  0.0500nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0680nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50114701(But-3-enoic acid {2-[5-methoxy-2-(3-methoxy-benzyl...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.174nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011344(CHEMBL3260982)
Affinity DataKi:  0.180nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.220nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM85066(Luzindole,5-Methoxy)
Affinity DataKi:  0.25nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.275nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011344(CHEMBL3260982)
Affinity DataKi:  0.290nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50114704(CHEMBL33549 | N-(2-(5-methoxy-2-(3-methoxybenzyl)b...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [125I]2-iodomelatonin from MT2 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086001(CHEMBL274438 | N-[2-(11-Methoxy-6,7-dihydro-5H-ben...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Rluc fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  0.600nMAssay Description:Agonist activity at MT2 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125757(CHEMBL14453 | N,N'-(2,2'-(7,7'-(butane-1,4-diylbis...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50149181(CHEMBL334079 | Cyclopropanecarboxylic acid {3-[2-(...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598933(CHEMBL5174929)
Affinity DataKi:  0.692nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to YFP fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM85054(1-[3-(5-Methoxy-1H-indol-3-yl)piperidino]ethanone ...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011353(CHEMBL3260987)
Affinity DataKi:  1.20nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in mouse NIH3T3 cells assessed as inhibition of forskolin-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011356(CHEMBL3260984)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to MT1 receptor (unknown origin) expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011349(CHEMBL189449)
Affinity DataKi:  1.30nMAssay Description:Antagonist activity at MT2 receptor (unknown origin) expressed in mouse NIH3T3 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598933(CHEMBL5174929)
Affinity DataKi:  1.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011338(CHEMBL3260979)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50114716(CHEMBL329263 | N-[2-(2-Benzyl-5-methoxy-benzofuran...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I]2-iodomelatonin from MT1 receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50340325(CHEMBL1760945 | N-(2-(6-Methoxy-1H-pyrrolo[2,3-b]p...)
Affinity DataKi:  1.40nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in HEK293 cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50240440(4-P-PDOT | CHEMBL285718 | N-(4-Phenyl-1,2,3,4-tetr...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataKi:  1.80nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598930(CHEMBL5173623)
Affinity DataKi:  2nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataKi:  2.20nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011338(CHEMBL3260979)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598930(CHEMBL5173623)
Affinity DataKi:  2.30nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125757(CHEMBL14453 | N,N'-(2,2'-(7,7'-(butane-1,4-diylbis...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011356(CHEMBL3260984)
Affinity DataKi:  3.40nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to YFP fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM82556(melatonin, 6-Methoxy)
Affinity DataKi:  3.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT2 receptor expressed in African green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50125754(CHEMBL429392 | N,N'-(2,2'-(7,7'-(propane-1,3-diylb...)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011354(CHEMBL3260985)
Affinity DataKi:  3.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50086013(CHEMBL10009 | N-[2-(2-Methoxy-6H-isoindolo[2,1-a]i...)
Affinity DataKi:  4.5nMAssay Description:Displacement of [125I]2-iodomelatonin from human recombinant MT1 receptor expressed in mouse NIH3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598931(CHEMBL5209359)
Affinity DataKi:  4.60nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes under dark condition by radi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011351(CHEMBL1097525)
Affinity DataKi:  5.20nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to Rluc fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1B(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598932(CHEMBL5195595)
Affinity DataKi:  6.90nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT2 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

Target5-hydroxytryptamine receptor 4(Human)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50219133(2-[4-({5-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50598932(CHEMBL5195595)
Affinity DataKi:  7.80nMAssay Description:Displacement of 2-[125I]iodomelatonin from human melatonin MT1 receptor stably expressing in human HEK293 cell membranes in presence of light-activat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelatonin receptor type 1A(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50011355(CHEMBL3260986)
Affinity DataKi:  7.90nMAssay Description:Displacement of [125I]2-iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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