Compile Data Set for Download or QSAR
Report error Found 4434 with Last Name = 'jones' and Initial = 'g'
LigandPNGBDBM762547(2-[[6-(5-amino-4-methyl-3-pyridyl)-7-fluoro-3- iso...)
Affinity DataKi:  0.0100nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762563(tert-butyl 7-[7-fluoro-3-[(6-methyl-7-oxo-5,8- dih...)
Affinity DataKi:  0.0100nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762584(1H-pyrido[2,3-b][1,4]oxazin-7-yl)isoquinolin- | US...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762697((S)-7-(3-((5,6-dihydro-11H-imidazo[1,2- | US123782...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762585((S)-2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- | US1...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762586(pyrido[2,3-b][1,4]oxazin-7-yl)isoquinolin-3- | US1...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762699(2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- | US12378...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762605(2-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoq...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762669(2'-((6-(5-amino-4-methylpyridin-3-yl)-8- fluoroiso...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762604(N-(6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoqu...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762668(2'-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroiso...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762590(N-(7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,3...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762625(N-(7-fluoro-6-(9-methyl-1,2,3,4- tetrahydropyrido[...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762579(N-(7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,3...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762596(2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762581(2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762647((R)-2'-((7-fluoro-6-(8-hydroxy-4-methyl- | US12378...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762648(5,6,7,8-tetrahydro-1,5-naphthyridin-3- | US1237824...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762573(2-((7,8-difluoro-6-(8-methyl-2,3-dihydro-1H- pyrid...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762606(2-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoq...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762609(fluoroisoquinolin-3-yl)amino)-6-(tert-butyl)-4- | ...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762601(2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,...)
Affinity DataKi:  0.0130nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762551(2-((7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762583((S)-2-(2-((7-fluoro-6-(8-methyl-2,3-dihydro- | US1...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762594((S)-2-(2-((6-(5-amino-4-methylpyridin-3-yl)-7- | U...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762598(N-(6-(5-amino-4-methylpyridin-3-yl)-7,8- difluoroi...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762602(N-(7,8-difluoro-6-(8-methyl-2,3-dihydro-1H- pyrido...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762692(2-((7-fluoro-6-(4,7,7-trimethyl-8-oxo-5,6,7,8- tet...)
Affinity DataKi:  0.0140nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762600(2-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoq...)
Affinity DataKi:  0.0150nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762676(5,6,7,8-tetrahydro-1,5-naphthyridin-3- | US1237824...)
Affinity DataKi:  0.0160nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762597(2-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoq...)
Affinity DataKi:  0.0170nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762634(2-((7-fluoro-6-(4-methyl-5,6,7,8-tetrahydro- 1,5-n...)
Affinity DataKi:  0.0180nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762577(pyrido[2,3-b][1,4]oxazin-7-yl)isoquinolin-3- | US1...)
Affinity DataKi:  0.0180nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762626(2-((6-(3,8-dimethyl-2,3-dihydro-1H- pyrido[2,3-b][...)
Affinity DataKi:  0.0180nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762588(fluoroisoquinolin-3-yl)amino)-6-(1- | US12378249, ...)
Affinity DataKi:  0.0190nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM503879(1-[3-[4-[[8-amino-6-(4-methyl-3-pyridyl)- 2,7-naph...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM762567(2-[[7-fluoro-6-(8-methyl-2,3-dihydro-1H- pyrido[2,...)
Affinity DataKi:  0.0200nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM503863(trans-N-[8-amino-6-(4-methyl-3-pyridyl)- 2,7-napht...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM503914((1S,2S)-N-(8-amino-5-fluoro-6-(4- methylpyridin-3-...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM504044(US11034692, Compound 313)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM504062((1R,2R)-N-(8-amino-6-(4-methylpyridin- 3-yl)-2,7-n...)
Affinity DataKi: <0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM762698(alpyrazolo[1,5-d][1,4]diazepin-8-yl)amino)-7- | US...)
Affinity DataKi:  0.0200nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM504049((1R,2S)—N-(8-amino-5-cyclopropyl-6-(4-methylp...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM762652(2-((6-(8,8-difluoro-4-methyl-5,6,7,8- tetrahydro-1...)
Affinity DataKi:  0.0200nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM504051((1S,2S)—N-(8-amino-6-(4-methyl-2-phenylpyridi...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM503940(1-(3-(4-(8-amino-6-(4-methylpyridin-3- yl)-2,7-nap...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM503988(2-[[8-amino-6-(4-methylpyridin-3-yl)-2,7- naphthyr...)
Affinity DataKi:  0.0200nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM503999(3-[[8-Amino-6-(4-methylpyridin-3-yl)-2,7- naphthyr...)
Affinity DataKi:  0.0210nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM503978(US11034692, Compound 247)
Affinity DataKi:  0.0220nMAssay Description:Lanth: For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. Th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2021
Entry Details
US Patent

LigandPNGBDBM762599(2-((6-(5-amino-4-methylpyridin-3-yl)-7- fluoroisoq...)
Affinity DataKi:  0.0230nMAssay Description:Assay Condition:The following assay concentrations and times were used: 2 nM HPK1, 2 nM Eu-Anti-GST Ab, and 15 nM Tracer222, with 60 min incubation t...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

Displayed 1 to 50 (of 4434 total ) | Next | Last >>
Jump to: