Compile Data Set for Download or QSAR
Report error Found 31 with Last Name = 'kagabu' and Initial = 's'
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50: 20nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488029((S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 190nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488030((R,S)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 210nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50251867(N-(3-((6-chloropyridin-3-yl)methyl)thiazol-2(3H)-y...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50251868({(2Z)-3-[(6-chloropyridin-3-yl)methyl]-1,3-thiazol...)
Affinity DataIC50: 860nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50252631(N-(3-((6-chloropyridin-3-yl)methyl)thiazol-2(3H)-y...)
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50488028((R)-METHYL-IMIDACLOPRID)
Affinity DataIC50: 950nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143314(CHEMBL298826 | (+)-Epibatidine | 2-(6-Chloro-pyrid...)
Affinity DataIC50: 1.34E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50143320(2-(6-Chloro-pyridin-3-yl)-7-aza-bicyclo[2.2.1]hept...)
Affinity DataIC50: 2.79E+3nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataIC50: 1.19E+4nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM82068(Nicotine-D salicylate | CHEMBL9732 | Nicotine-L sa...)
Affinity DataIC50: 4.22E+5nMAssay Description:Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
University of California

Curated by ChEMBL
LigandPNGBDBM50095649((2E)-1-[(5-azido-6-chloropyridin-3-yl)methyl]-N-ni...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487224(CHEMBL2252498)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rat)
University of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  50nMAssay Description:Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487219(CHEMBL2252497)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487229(CHEMBL2252496)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487226(CHEMBL2252501)
Affinity DataKi:  800nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487222(CHEMBL2252352)
Affinity DataKi:  1.46E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487231(CHEMBL2252353)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487227(CHEMBL447459)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487225(CHEMBL2252499)
Affinity DataKi:  2.30E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487223(CHEMBL2252495)
Affinity DataKi:  2.66E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487232(CHEMBL2252503)
Affinity DataKi:  2.77E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487220(CHEMBL2252350)
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487233(CHEMBL2252500)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487228(CHEMBL2252504)
Affinity DataKi:  1.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487230(CHEMBL2252502)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487221(CHEMBL2252351)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNicotinic acetylcholine receptor alpha 5 subunit(House fly)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50487218(CHEMBL2252349)
Affinity DataKi:  2.60E+4nMAssay Description:Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed