Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 108 with Last Name = 'kakefuda' and Initial = 'a'
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108501(2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimet...)
Affinity DataKi:  0.102nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.620nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  0.770nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]-AVP on rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114033(CHEMBL86667 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  1.01nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114028(1-{6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  1.04nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114034(1'-{6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-...)
Affinity DataKi:  1.05nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  1.19nMAssay Description:Binding affinity at cloned human Vasopressin V2 receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108498(Biphenyl-2-carboxylic acid (4-{5-[2-(4-dimethylami...)
Affinity DataKi:  1.20nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  1.43nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114025(4-{4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  2.12nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108493(2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']...)
Affinity DataKi:  2.90nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114032(CHEMBL86577 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  3.03nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114045(1-{5-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  4.09nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114038(1-{7-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108494(2-Methyl-furan-3-carboxylic acid (4-{[2-(6-[1,4']b...)
Affinity DataKi:  5nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108495(1N-methyl-1N-{4-methyl-2-[6-(4-methylhexahydro-1-p...)
Affinity DataKi:  5.70nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108499(1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-p...)
Affinity DataKi:  7.60nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114037(4-{3-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  7.84nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114041(CHEMBL316093 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,...)
Affinity DataKi:  8.09nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108500(2-Methyl-furan-3-carboxylic acid [4-(methyl-{4-met...)
Affinity DataKi:  8.80nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114043(3-Biphenyl-4-yl-4-[2-(6-imidazol-1-yl-hexyloxy)-ph...)
Affinity DataKi:  9.06nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114040(6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4-yl...)
Affinity DataKi:  9.16nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114034(1'-{6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-...)
Affinity DataKi:  9.69nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114029(1-{8-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  13.2nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114039(1-{6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  13.9nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114028(1-{6-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  17.3nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  23.5nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  24nMAssay Description:Evaluated for the binding affinity towards Vasopressin V1a receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114026(1-{4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  29.1nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114033(CHEMBL86667 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  32.4nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108501(2-Methyl-furan-3-carboxylic acid (4-{5-[2-(4-dimet...)
Affinity DataKi:  34nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114042(1-{3-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  38.3nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114036(1-{10-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-...)
Affinity DataKi:  39.4nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108493(2-Methyl-furan-3-carboxylic acid [4-({2-[4-([1,4']...)
Affinity DataKi:  42nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114044(4-{2-[2-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  55.5nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114032(CHEMBL86577 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  62.7nMAssay Description:Binding affinity at Vasopressin V1a receptor, performed using [3H]-AVP on rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108500(2-Methyl-furan-3-carboxylic acid [4-(methyl-{4-met...)
Affinity DataKi:  73nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366798(CHEMBL1794053)
Affinity DataKi:  79nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108494(2-Methyl-furan-3-carboxylic acid (4-{[2-(6-[1,4']b...)
Affinity DataKi:  95nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114035(3-Biphenyl-4-yl-4-(2-methoxy-phenyl)-5-methyl-4H-[...)
Affinity DataKi:  120nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50366798(CHEMBL1794053)
Affinity DataKi:  168nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  178nMAssay Description:Binding affinity at cloned human Vasopressin V2 receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114046(1-{6-[3-(3-Biphenyl-4-yl-5-methyl-[1,2,4]triazol-4...)
Affinity DataKi:  214nMAssay Description:Binding affinity at cloned human Vasopressin V1a receptor stably expressed in CHO cells, using [3H]-AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114031((2S)-1-[(2R,3S)-5-chloro-3-(2-chlorophenyl)-1-(3,4...)
Affinity DataKi:  285nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]-AVP on rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108497(2-Methyl-furan-3-carboxylic acid (4-{[4'-([1,4']bi...)
Affinity DataKi:  335nMAssay Description:Evaluated for the binding affinity towards vasopressin (V1A) receptor in rat liver membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50114032(CHEMBL86577 | {4-[2-(3-Biphenyl-4-yl-5-methyl-[1,2...)
Affinity DataKi:  364nMAssay Description:Binding affinity at Vasopressin V2 receptor, performed using [3H]-AVP on rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Yamanouchi Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50108499(1N-methyl-1N-{4-methyl-2-[4-(4-methylhexahydro-1-p...)
Affinity DataKi:  445nMAssay Description:Evaluated for the binding affinity towards vasopressin (V2) receptor in rat kidney membrane using [3H]AVP as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 108 total ) | Next | Last >>
Jump to: