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TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157484(4-(1-benzyl-7-chloro-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataEC50:  390nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157486(4-(6-HYDROXY-1H-INDAZOL-3-YL)BENZENE-1,3-DIOL | CH...)
Affinity DataEC50:  298nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157487(4-(6-hydroxy-1-propyl-1H-indazol-3-yl)benzene-1,3-...)
Affinity DataEC50:  1.22E+3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157488(4-(7-chloro-1-cyclopentyl-1H-indazol-3-yl)phenol |...)
Affinity DataEC50:  98nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157489(4-[1-(3-fluorophenyl)-6-hydroxy-1H-indazol-3-yl]be...)
Affinity DataEC50:  140nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157483(4-(1-cyclopentyl-7-fluoro-1H-indazol-3-yl)phenol |...)
Affinity DataEC50:  330nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157485(4-[1-isopropyl-7-(trifluoromethyl)-1H-indazol-3-yl...)
Affinity DataEC50:  11nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157499(4-(1-methyl-6-hydroxy-1H-indazol-3-yl)benzene-1,3-...)
Affinity DataEC50:  3.72E+3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157494(4-(1-butyl-6-hydroxy-1H-indazol-3-yl)benzene-1,3-d...)
Affinity DataEC50:  549nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157503(4-(7-methyl-1-propyl-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataEC50:  303nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157500(4-[6-hydroxy-1-(4-methylphenyl)-1H-indazol-3-yl]be...)
Affinity DataEC50:  149nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157497(4-[6-hydroxy-1-(2,2,2-trifluoroethyl)-1H-indazol-3...)
Affinity DataEC50:  4.79E+3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157495(4-(1-ethyl-6-hydroxy-1H-indazol-3-yl)benzene-1,3-d...)
Affinity DataEC50:  3.07E+3nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157498(4-(1-butyl-7-chloro-1H-indazol-3-yl)phenol | CHEMB...)
Affinity DataEC50:  63nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50157502(4-(7-chloro-1-propyl-1H-indazol-3-yl)phenol | CHEM...)
Affinity DataEC50:  138nMAssay Description:Activity at human ERalpha expressed in HAECT1 cells assessed as stimulation of creatine kinase activityMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168331(3-(2-Fluoro-4-hydroxy-phenyl)-7-hydroxy-naphthalen...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168341(7-(3-Fluoro-4-hydroxy-phenyl)-3-hydroxy-naphthalen...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168367(1-Chloro-8-fluoro-6-(4-hydroxy-phenyl)-naphthalen-...)
Affinity DataIC50: 1.10nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154088(7-bromo-2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 7...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168321(1-Chloro-6-(2-fluoro-4-hydroxy-phenyl)-naphthalen-...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168352(4-Ethynyl-6-(3-fluoro-4-hydroxy-phenyl)-naphthalen...)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154078(7-bromo-2-(4-hydroxy-2-methylphenyl)benzo[d]oxazol...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154134(2-(4-Hydroxy-phenyl)-7-propenyl-benzooxazol-5-ol |...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154137(3-(6-hydroxynaphthalen-2-yl)benzo[d]isoxazol-6-ol ...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154059(7-Bromo-2-(2-fluoro-4-hydroxy-phenyl)-benzooxazol-...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168347(6-(2-Chloro-4-hydroxy-phenyl)-naphthalen-2-ol | CH...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154048(3-(5-hydroxynaphthalen-1-yl)benzo[d]isoxazol-6-ol ...)
Affinity DataIC50: 1.5nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168358(8-Fluoro-6-(3-fluoro-4-hydroxy-phenyl)-naphthalen-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168353(8-Fluoro-6-(4-hydroxy-phenyl)-naphthalen-2-ol | CH...)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Mouse)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154088(7-bromo-2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 7...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to mouse ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM20731(4-bromo-6-(6-hydroxy-1,2-benzoxazol-3-yl)benzene-1...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154140(2-(2-fluoro-4-hydroxyphenyl)-7-vinylbenzo[d]oxazol...)
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154088(7-bromo-2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 7...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM20734(CHEMBL362307 | 4-chloro-6-(6-hydroxy-1,2-benzoxazo...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154084(7-bromo-2-(3-fluoro-4-hydroxyphenyl)benzo[d]oxazol...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168350(6-(2-Fluoro-4-hydroxy-phenyl)-naphthalen-2-ol | CH...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168335(3-Hydroxy-7-(4-hydroxy-phenyl)-naphthalene-1-carbo...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168386(7-(3-Fluoro-4-hydroxy-phenyl)-3-hydroxy-naphthalen...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Rat)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154057(2-(4-hydroxyphenyl)benzo[d]oxazol-5-ol | 2-(4-Hydr...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to rat ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154132(2-(2,6-Difluoro-4-hydroxy-phenyl)-7-vinyl-benzooxa...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor(Mouse)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to mouse ER alpha expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168365(3-(2,6-Difluoro-4-hydroxy-phenyl)-7-hydroxy-naphth...)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Mouse)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM17292([2,4,6,7-3H]-17beta-estradiol | [3H]-estradiol | 1...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to mouse ER beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168333(6-(2,6-Difluoro-4-hydroxy-phenyl)-naphthalen-2-ol ...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168354(7-Hydroxy-3-(4-hydroxy-phenyl)-naphthalene-1-carbo...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168384(8-Chloro-6-(4-hydroxy-phenyl)-naphthalen-2-ol | CH...)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50154064(2-(2-fluoro-4-hydroxyphenyl)-5-hydroxybenzo[d]oxaz...)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory concentration against human ER beta expressed in Escherichia coli was determined using [3H]17-beta-estradiol as radio ligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50168342(8-Ethyl-6-(3-fluoro-4-hydroxy-phenyl)-naphthalen-2...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of [3H]17-beta-estradiol binding to human estrogen receptor beta expressed in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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