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TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377933(CHEMBL1744354)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242595(CHEMBL487860 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242577(6-{[2-({2-[(2S,4S)-2-Cyano-4-fluoropyrrolidin-1-yl...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242517((2S,4S)-1-(N-Cyclopentylglycyl)-4-fluoropyrrolidin...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242576((2S,4S)-1-(N-{2-[(5-Chloropyridin-2-yl)amino]ethyl...)
Affinity DataIC50:  2.70nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242575((2S,4S)-4-Fluoro-1-{N-[2-(pyridin-2-ylamino)ethyl]...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242495((2S,4S)-1-[N-(tert-Butyl)glycyl]-4-fluoropyrrolidi...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242593(CHEMBL488036 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35718(benzazepine derivative, 20)
Affinity DataIC50:  3nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataIC50:  3nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242530((2S,4S)-1-(N-2-Adamantylglycyl)-4-fluoropyrrolidin...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242516((2S,4S)-1-(N-Cyclobutylglycyl)-4-fluoropyrrolidine...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242531((2S,4S)-4-Fluoro-1-[N-(3-hydroxy-1-adamantyl)-glyc...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242519((2S,4S)-1-(N-Cyclooctylglycyl)-4-fluoropyrrolidine...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242518((2S,4S)-4-Fluoro-1-{N-[1-(hydroxymethyl)cyclopenty...)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242529((2S,4S)-1-(N-1-Adamantylglycyl)-4-fluoropyrrolidin...)
Affinity DataIC50:  4.10nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242579(CHEMBL488418 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242513((2S,4S)-4-Fluoro-1-[N-(2-hydroxy-1,1-dimethylethyl...)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35725(benzazepine derivative, 34)
Affinity DataIC50:  5nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35719(benzazepine derivative, 21)
Affinity DataIC50:  5nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242533((2S,4S)-4-Fluoro-1-[N-(5-hydroxy-2-adamantyl)-glyc...)
Affinity DataIC50:  5.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242580(CHEMBL488419 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242594(CHEMBL519585 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242596(CHEMBL487861 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242476(CHEMBL471088 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  6.20nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35725(benzazepine derivative, 34)
Affinity DataIC50:  7nMAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM11113(6-{[2-({2-[(2S)-2-cyanopyrrolidin-1-yl]-2-oxoethyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35715(benzazepine derivative, 13a)
Affinity DataIC50:  7nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242475(CHEMBL470893 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242496((2S,4S)-4-Fluoro-1-(N-isopropylglycyl)pyrrolidine-...)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35721(benzazepine derivative, 30)
Affinity DataIC50:  8nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242578(CHEMBL487681 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242532((2S,4S)-4-Fluoro-1-[N-(3-methoxy-1-adamantyl)-glyc...)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242478((2S,4S)-4-Fluoro-1-{N-[1-(2-furyl)-1-methylethyl]-...)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242497((2S,4S)-4-Fluoro-1-[N-(3-isopropoxypropyl)glycyl]p...)
Affinity DataIC50:  8.70nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35720(benzazepine derivative, 22)
Affinity DataIC50:  9nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataIC50:  12nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242491((2S,4S)-4-Fluoro-1-{N-[1-methyl-1-(2-thienyl)-ethy...)
Affinity DataIC50:  12nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataIC50:  12nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377932(CHEMBL1203962)
Affinity DataIC50:  13nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242597(CHEMBL487862 | N-[2-({2-[(2S,4S)-2-Cyano-4-fluorop...)
Affinity DataIC50:  13nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052948(CHEMBL324251 | N-{4-[5-(Carbamoylmethyl-methyl-ami...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052924(2,4-Dichloro-N-[4-(5-dimethylamino-2,3,4,5-tetrahy...)
Affinity DataIC50:  13nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35724(benzazepine derivative, 33)
Affinity DataIC50:  13nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052930(2-Methyl-N-[4-(5-methyl-2,3,4,5-tetrahydro-benzo[b...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052925(CHEMBL331098 | N-[4-(5-Dimethylamino-2,3,4,5-tetra...)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Human)
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50242493((2S,4S)-1-{N-[(2E)-1,1-Dimethyl-3-phenylprop-2-en-...)
Affinity DataIC50:  16nMAssay Description:Inhibition of DPP4 in human plasma by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35718(benzazepine derivative, 20)
Affinity DataIC50:  17nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50052954(2-Methyl-N-[4-(2,3,4,5-tetrahydro-benzo[b]azepine-...)
Affinity DataIC50:  18nMAssay Description:Displacement of [3H]-AVP from its AVP-V2 receptor binding site in rat kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

LigandPNGBDBM35716(benzazepine derivative, 18)
Affinity DataIC50:  18nMpH: 7.4 T: 4°CAssay Description:After reaching confluence in 12-well or 24-well dishes, the cells were washed twice with ice-cold PBS and incubated for 2 hr with [3H]-AVP at 4 deg C...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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