Compile Data Set for Download or QSAR
maximum 50k data
Found 161 with Last Name = 'kortum' and Initial = 'sw'
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302437(3-(3-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-eth...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302449((2R,5S)-1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-...)
Affinity DataKi:  4nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302452((2S,4S)-1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302457(3-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-ethylt...)
Affinity DataKi:  8nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302437(3-(3-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-eth...)
Affinity DataKi:  10nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302459((R)-biphenyl-4-yl(4-(2-(2,3-dihydroxypropylamino)-...)
Affinity DataKi:  19nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302449((2R,5S)-1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-...)
Affinity DataKi:  21nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302451(CHEMBL568566 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  27nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302434(CHEMBL585852 | biphenyl-4-yl(4-(6-ethylthieno[2,3-...)
Affinity DataKi:  29nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302452((2S,4S)-1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-...)
Affinity DataKi:  31nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302453(1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-ethylt...)
Affinity DataKi:  31nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302458(CHEMBL585948 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  35nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302446(3-(3-(6-ethyl-4-(4-isobutyrylpiperazin-1-yl)thieno...)
Affinity DataKi:  36nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302454(CHEMBL565618 | biphenyl-4-yl(4-(6-ethyl-2-(2-hydro...)
Affinity DataKi:  37nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302444(3-(3-(6-ethyl-4-(4-(5-phenylpicolinoyl)piperazin-1...)
Affinity DataKi:  37nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302446(3-(3-(6-ethyl-4-(4-isobutyrylpiperazin-1-yl)thieno...)
Affinity DataKi:  46nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302441(3-(3-(4-(4-(2-(3,4-difluorophenyl)acetyl)piperazin...)
Affinity DataKi:  68nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302459((R)-biphenyl-4-yl(4-(2-(2,3-dihydroxypropylamino)-...)
Affinity DataKi:  75nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302450(CHEMBL585317 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  78nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302457(3-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-ethylt...)
Affinity DataKi:  122nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302432(CHEMBL566447 | naphthalen-1-yl 4-(6-ethylthieno[2,...)
Affinity DataKi:  130nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302441(3-(3-(4-(4-(2-(3,4-difluorophenyl)acetyl)piperazin...)
Affinity DataKi:  140nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302444(3-(3-(6-ethyl-4-(4-(5-phenylpicolinoyl)piperazin-1...)
Affinity DataKi:  161nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302454(CHEMBL565618 | biphenyl-4-yl(4-(6-ethyl-2-(2-hydro...)
Affinity DataKi:  163nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302442(3-(3-(6-ethyl-4-(4-(3,3,3-trifluoropropanoyl)piper...)
Affinity DataKi:  172nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302442(3-(3-(6-ethyl-4-(4-(3,3,3-trifluoropropanoyl)piper...)
Affinity DataKi:  177nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302443(3-(3-(6-ethyl-4-(4-(2-(3-methoxyphenoxy)acetyl)pip...)
Affinity DataKi:  191nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302453(1-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-ethylt...)
Affinity DataKi:  203nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302438(3-(3-(6-ethyl-4-(4-(3-phenoxypropanoyl)piperazin-1...)
Affinity DataKi:  213nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302447(3-(3-(6-ethyl-4-(4-(2-phenylacetyl)piperazin-1-yl)...)
Affinity DataKi:  223nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302447(3-(3-(6-ethyl-4-(4-(2-phenylacetyl)piperazin-1-yl)...)
Affinity DataKi:  231nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302456((4-(2-(4-aminopiperidin-1-yl)-6-ethylthieno[2,3-d]...)
Affinity DataKi:  240nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302458(CHEMBL585948 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  241nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302440(3-(3-(6-ethyl-4-(4-propionylpiperazin-1-yl)thieno[...)
Affinity DataKi:  295nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302451(CHEMBL568566 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  297nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302456((4-(2-(4-aminopiperidin-1-yl)-6-ethylthieno[2,3-d]...)
Affinity DataKi:  325nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302440(3-(3-(6-ethyl-4-(4-propionylpiperazin-1-yl)thieno[...)
Affinity DataKi:  367nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302439(3-(3-(4-(4-acetylpiperazin-1-yl)-6-ethylthieno[2,3...)
Affinity DataKi:  380nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302448(CHEMBL566037 | biphenyl-4-yl(4-(6-ethyl-2-(piperaz...)
Affinity DataKi:  397nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302448(CHEMBL566037 | biphenyl-4-yl(4-(6-ethyl-2-(piperaz...)
Affinity DataKi:  410nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302450(CHEMBL585317 | biphenyl-4-yl(4-(6-ethyl-2-(3-hydro...)
Affinity DataKi:  441nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302443(3-(3-(6-ethyl-4-(4-(2-(3-methoxyphenoxy)acetyl)pip...)
Affinity DataKi:  447nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302439(3-(3-(4-(4-acetylpiperazin-1-yl)-6-ethylthieno[2,3...)
Affinity DataKi:  460nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302445(3-(3-(6-ethyl-4-(4-(2-phenoxyacetyl)piperazin-1-yl...)
Affinity DataKi:  539nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302445(3-(3-(6-ethyl-4-(4-(2-phenoxyacetyl)piperazin-1-yl...)
Affinity DataKi:  593nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302431(1-(4-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperazin...)
Affinity DataKi:  660nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302438(3-(3-(6-ethyl-4-(4-(3-phenoxypropanoyl)piperazin-1...)
Affinity DataKi:  783nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302455(1-(4-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-eth...)
Affinity DataKi:  839nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302455(1-(4-(4-(4-(biphenylcarbonyl)piperazin-1-yl)-6-eth...)
Affinity DataKi:  1.81E+3nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed in CHO cell membrane in presence of HSA and human AGPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50302433(1-(4-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperazin...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity to human recombinant P2Y12 receptor expressed on CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 161 total ) | Next | Last >>
Jump to: