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TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataKi:  0.430nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  2.60nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
PDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273464((1S,9S,10S)-11-(2-phenylethyl)-8-oxa-11-azatetracy...)
Affinity DataKi:  7nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V2 receptor(Human)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM35714(CHEMBL420762 | Mozavaptan | N-[4-(5-Dimethylamino-...)
Affinity DataKi:  9.42nMAssay Description:Concentration of the compound which inhibit [3H]-AVP binding to human Vasopressin V2 receptor coded HeLa cells by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetVasopressin V1a receptor(Rat)
Otsuka Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50029644(CHEMBL296908 | N-(3-(4-(4-(2-oxo-3,4-dihydroquinol...)
Affinity DataKi:  32nMAssay Description:Binding affinity of the compound towards Vasopressin V1a receptor in rat liverMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  42nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  78nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348870(CHEMBL1808302)
Affinity DataKi:  98nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  102nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348869(CHEMBL1808300)
Affinity DataKi:  167nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348869(CHEMBL1808300)
Affinity DataKi:  171nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348871(CHEMBL1808303)
Affinity DataKi:  199nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273414((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348871(CHEMBL1808303)
Affinity DataKi:  250nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  352nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348872(CHEMBL1808304)
Affinity DataKi:  367nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348872(CHEMBL1808304)
Affinity DataKi:  384nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348870(CHEMBL1808302)
Affinity DataKi:  486nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273416((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273414((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  560nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273415((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi:  620nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  740nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273934((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-methyl-1...)
Affinity DataKi:  910nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273416((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  1.22E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273416((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  2.53E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273415((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi:  2.78E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348868(CHEMBL1808301)
Affinity DataKi: >2.80E+3nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50348867(CHEMBL1808299)
Affinity DataKi: >2.80E+3nMAssay Description:Displacement of [125I]IOXY from human mu opioid receptor expressed in CHO cells coexpressing human recombinant MOR after 2 hrs by liquid scintillatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273414((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-pheneth...)
Affinity DataKi:  2.84E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273415((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi: >2.93E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273934((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-methyl-1...)
Affinity DataKi:  3.21E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273413((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi:  3.43E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  3.71E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi:  4.76E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273413((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi:  4.82E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348869(CHEMBL1808300)
Affinity DataKi: >4.90E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348870(CHEMBL1808302)
Affinity DataKi: >4.90E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348868(CHEMBL1808301)
Affinity DataKi: >4.90E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348867(CHEMBL1808299)
Affinity DataKi: >4.90E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348872(CHEMBL1808304)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348871(CHEMBL1808303)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273933((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273935((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-phenethy...)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [125I]IOXY from human delta opioid receptor expressed in CHO cells coexpressing human recombinant DOR after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348867(CHEMBL1808299)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMu-type opioid receptor(Human)
National Institute On Drug Abuse and The National Institute On Alcohol Abuse and Alcoholism

Curated by ChEMBL
LigandPNGBDBM50273413((3R*,6aS*,11aR*)-1,3,4,5,6,11a-Hexahydro-2-methyl-...)
Affinity DataKi: >8.00E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetKappa-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50348868(CHEMBL1808301)
Affinity DataKi: >8.60E+3nMAssay Description:Displacement of [125I]IOXY from human kappa opioid receptor expressed in CHO cells coexpressing human recombinant KOP after 2 hrs by liquid scintilla...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetDelta-type opioid receptor(Human)
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50273934((4R*,6aS*,11bR*)-2,3,4,5,6,6a-Hexahydro-3-methyl-1...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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