TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 25nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 33nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 36nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 45nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 47nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 49nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 79nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 84nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 96nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 101nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 115nMAssay Description:Antagonist activity at human MCHR1 expressed in CHO-K1 cells assessed as inhibition of MCH peptide mediated response measuring [3H]inositol phosphate...More data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Dr. Reddy's Laboratories Ltd
Curated by ChEMBL
Affinity DataIC50: 116nMAssay Description:Displacement of [125I]MCH from human recombinant MCHR1 expressed in CHO-K1 cell membranes after 2 hrs by SPA binding assayMore data for this Ligand-Target Pair
