Compile Data Set for Download or QSAR
Found 184 with Last Name = 'lecis' and Initial = 'd'
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita degli Studi di Milano

LigandPNGBDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
Affinity DataKi:  25nM ΔG°:  -43.1kJ/mole IC50:  460nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 3(Homo sapiens (Human))
Universita degli Studi di Milano

LigandPNGBDBM13212((3S,6S,9aS)-N-(diphenylmethyl)-6-[(2S)-2-(methylam...)
Affinity DataKi:  61nM ΔG°:  -40.9kJ/mole IC50:  530nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Milano

LigandPNGBDBM26205((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(2-ami...)
Affinity DataKi:  220nM ΔG°:  -37.6kJ/mole IC50:  250nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Milano

LigandPNGBDBM26203((3S,6S,7S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphe...)
Affinity DataKi:  250nM ΔG°:  -37.3kJ/mole IC50:  270nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Milano

LigandPNGBDBM13211((3S,6S,9aS)-6-[(2S)-2-aminobutanamido]-N-(diphenyl...)
Affinity DataKi:  420nM ΔG°:  -36.0kJ/mole IC50:  460nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
University of Milano

LigandPNGBDBM26204((3S,6S,7R,9aS)-6-[(2S)-2-aminobutanamido]-7-(amino...)
Affinity DataKi:  870nM ΔG°:  -34.2kJ/mole IC50:  970nMpH: 7.5 T: 2°CAssay Description:Fluorescence polarization was measured on an Ultra plate reader (Tecan) at excitation and emission wavelengths of 485 and 530 nm, respectively. The e...More data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401475(CHEMBL2205248)
Affinity DataIC50:  1.10nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50240586(CHEMBL4098982)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401483(CHEMBL2204574)
Affinity DataIC50:  1.40nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401484(CHEMBL2204575)
Affinity DataIC50:  1.40nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50240587(CHEMBL4070316)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM32609(1-aza-2-oxobicyclo[5.3.0]decane scaffold, 36b)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401493(CHEMBL2205246)
Affinity DataIC50:  1.5nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401477(CHEMBL2204567)
Affinity DataIC50:  1.5nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50240589(CHEMBL4091245)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401489(CHEMBL2204580)
Affinity DataIC50:  1.60nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401485(CHEMBL2204576)
Affinity DataIC50:  1.70nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50240592(CHEMBL4097534)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of SMAC derived peptide abuRPF-K(5-Fam)-NH2 interaction with recombinant human C-terminal 6His-tagged cIAP1 BIR3 domain (245 to 357 residu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401481(CHEMBL2204572)
Affinity DataIC50:  1.70nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401492(CHEMBL2204582)
Affinity DataIC50:  1.90nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365839(CHEMBL1957014)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365847(CHEMBL1957024)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365848(CHEMBL1957023)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365840(CHEMBL1957013)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365838(CHEMBL1957015)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365836(CHEMBL1957017)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365846(CHEMBL1957026)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365837(CHEMBL1957016)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365851(CHEMBL1957019)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365841(CHEMBL575256)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365845(CHEMBL1957105)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365835(CHEMBL1957018)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365844(CHEMBL1957106)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365849(CHEMBL1957021)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365843(CHEMBL1957107)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365850(CHEMBL1957020)
Affinity DataIC50: <2nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401488(CHEMBL2204579)
Affinity DataIC50:  2.30nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401474(CHEMBL2205247)
Affinity DataIC50:  2.60nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365842(CHEMBL1957022)
Affinity DataIC50:  2.60nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401482(CHEMBL2204573)
Affinity DataIC50:  2.90nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401487(CHEMBL2204578)
Affinity DataIC50:  3.20nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401479(CHEMBL2204569)
Affinity DataIC50:  3.20nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50365834(CHEMBL1957025)
Affinity DataIC50:  3.30nMAssay Description:Displacement of AbuRPF-K(5-Fam)-NH2 from human recombinant His-tagged-cIAP1 BIR3 domain after 3 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401480(CHEMBL2204571)
Affinity DataIC50:  3.30nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401488(CHEMBL2204579)
Affinity DataIC50:  3.5nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401487(CHEMBL2204578)
Affinity DataIC50:  3.80nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401483(CHEMBL2204574)
Affinity DataIC50:  3.90nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401476(CHEMBL2205249)
Affinity DataIC50:  4.40nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBaculoviral IAP repeat-containing protein 2(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401478(CHEMBL2204568)
Affinity DataIC50:  5nMAssay Description:Displacement of FITC-Smac from human recombinant His-tagged cIAP-1 BIR3 domain (245 to 357 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Fondazione IRCCS Istituto Nazionale dei Tumori

Curated by ChEMBL
LigandPNGBDBM50401490(CHEMBL2204570)
Affinity DataIC50:  5.30nMAssay Description:Displacement of Smac-1F from human His-tagged XIAP linker BIR2-BIR3 linker (124 to 356 residues) after 3 hrs by fluorescent polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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