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TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails PubMedPDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails PubMedPDB3D3D Structure (crystal)

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM21015((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  1.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM21025((2R)-2-[(2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydro...)
Affinity DataKi:  4.90nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50209301((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi:  16.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50044896(CHEMBL162564 | Morphiceptin | Tyr-Pro-D-Phe-Pro-NH...)
Affinity DataKi:  34.9nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50209301((S)-1-((S)-2-amino-3-(4-hydroxyphenyl)propanoyl)-N...)
Affinity DataKi:  37nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM50044896(CHEMBL162564 | Morphiceptin | Tyr-Pro-D-Phe-Pro-NH...)
Affinity DataKi:  63nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM21008((4S,7S,13S)-13-[(2S)-2-amino-3-(4-hydroxyphenyl)pr...)
Affinity DataKi:  490nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetMu-type opioid receptor(Rat)
Burroughs Wellcome

Curated by PDSP Ki Database
LigandPNGBDBM82064(CAS_79805-24-6 | NSC_16219643 | beta-Casomorphin)
Affinity DataKi:  1.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138201(US8871778, 144)
Affinity DataIC50:  0.700nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138204(US8871778, 161)
Affinity DataIC50:  0.700nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138200(US8871778, 141)
Affinity DataIC50:  1nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138210(US8871778, 189)
Affinity DataIC50:  1nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124868(CHEMBL3622958)
Affinity DataIC50:  1.70nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124761(CHEMBL3622935)
Affinity DataIC50:  1.90nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124705(CHEMBL3622924)
Affinity DataIC50:  2.30nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124709(CHEMBL3622928)
Affinity DataIC50:  3.5nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124756(CHEMBL3622934)
Affinity DataIC50:  3.70nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179403(US9126973, 8)
Affinity DataIC50:  4nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124765(CHEMBL3622938)
Affinity DataIC50:  5nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124707(CHEMBL3622926)
Affinity DataIC50:  5.40nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124807(CHEMBL3622944)
Affinity DataIC50:  5.70nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179422(US9126973, 19)
Affinity DataIC50:  6nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124711(CHEMBL3622930)
Affinity DataIC50:  6.20nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124816(CHEMBL3622945)
Affinity DataIC50:  6.30nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124710(CHEMBL3622929)
Affinity DataIC50:  7.30nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124771(CHEMBL3622940)
Affinity DataIC50:  7.30nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124839(CHEMBL3622946)
Affinity DataIC50:  7.90nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124869(CHEMBL3622960)
Affinity DataIC50:  8nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124806(CHEMBL3622943)
Affinity DataIC50:  8.90nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124866(CHEMBL3622953)
Affinity DataIC50:  9.20nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179375(US9126973, 1)
Affinity DataIC50:  12nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124781(CHEMBL3622942)
Affinity DataIC50:  12nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124763(CHEMBL3622936)
Affinity DataIC50:  13nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124778(CHEMBL3622941)
Affinity DataIC50:  14nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124769(CHEMBL3622939)
Affinity DataIC50:  17nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124764(CHEMBL3622937)
Affinity DataIC50:  18nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124865(CHEMBL3622951)
Affinity DataIC50:  20nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138203(US8871778, 160)
Affinity DataIC50:  20nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179408(US9126973, 10)
Affinity DataIC50:  21nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179418(US9126973, 15)
Affinity DataIC50:  23nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent


TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124867(CHEMBL3622954)
Affinity DataIC50:  23nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138221(US8871778, 52)
Affinity DataIC50:  37nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124708(CHEMBL3622927)
Affinity DataIC50:  38nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138200(US8871778, 141)
Affinity DataIC50:  38nMAssay Description:Inhibition of SYK-mediated TNFalpha production in human IgG-stimulated human THP1 cells incubated for 18 hrs by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedPDB3D3D Structure (crystal)

TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM50124713(CHEMBL3622932)
Affinity DataIC50:  39nMT: 25°CAssay Description:Inhibition of purified full-length human SYK pre-incubated for 30 mins at room temperature before Ulight-TK peptide substrate addition and measured 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetHematopoietic prostaglandin D synthase(Human)
Cayman Chemical

US Patent
LigandPNGBDBM179409(US9126973, 11)
Affinity DataIC50:  41nMpH: 8.0 T: 25°CAssay Description:The assay is carried out by the following steps: 1. Inhibitor screening is performed in 100 mM Tris-HCl, pH 8.0 containing 1 mM GSH, 1 mM MgCl.sub.2,...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetTyrosine-protein kinase SYK(Human)
Kangwon National University

Curated by ChEMBL
LigandPNGBDBM138210(US8871778, 189)
Affinity DataIC50:  44nMAssay Description:Inhibition of SYK-mediated TNFalpha production in human IgG-stimulated human THP1 cells incubated for 18 hrs by ELISA methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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