Compile Data Set for Download or QSAR
Found 127 with Last Name = 'lezoualc''h' and Initial = 'f'
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.0780nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4D receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4A receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4C receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to Rluc fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4B receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29525(3H-GR113808 | CHEMBL518682 | GR 113808 | [3H] GR 1...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to YFP fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092543(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  1nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092551(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(2,3,5,6...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092547(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrid...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092550(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrid...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50293279(1-Methyl-5-[(1-propylpiperidin-4-yl)methyloxy]-pyr...)
Affinity DataKi:  1.74nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092546(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(6-ch...)
Affinity DataKi:  2nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092543(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  2.47nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4C receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50108392((3-ENDO)-8-METHYL-8-AZABICYCLO[3.2.1]OCT-3-YL 1H-I...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity at 5HT3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092545(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(3-me...)
Affinity DataKi:  3nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174419(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  3nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to YFP fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092548(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrid...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092543(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4A receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  3.69nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4D receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174414(4-(3-{1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbon...)
Affinity DataKi:  5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174432(1-[2-(3-amino-4-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174440(1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)...)
Affinity DataKi:  5nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50413548(CHEMBL512679)
Affinity DataKi:  5.37nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5.60nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  5.70nMAssay Description:Binding affinity to Rluc fused 5HT4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174416(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  6nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50413547(CHEMBL448702)
Affinity DataKi:  6.46nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174434(1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)...)
Affinity DataKi:  7nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50219133(2-[4-({5-[(1-{2-[(4-amino-5-chloro-2-methoxyphenyl...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092543(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  7.03nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4D receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  7.98nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4C receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174421(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  8nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174430(1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)...)
Affinity DataKi:  8nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092543(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  8.10nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4B receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  8.40nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4A receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50413546(CHEMBL513254)
Affinity DataKi:  8.51nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50413545(CHEMBL469575)
Affinity DataKi:  8.71nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174435(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  9nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174420(1-[2-(4-amino-5-chloro-2-hydroxyphenylcarbonyloxy)...)
Affinity DataKi:  9nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174431(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]GR-113808 from human 5HT4e receptor expressed in C6 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092555(4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-pyrim...)
Affinity DataKi:  9.20nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Université de Caen

Curated by ChEMBL
LigandPNGBDBM50413544(CHEMBL511794)
Affinity DataKi:  9.55nMAssay Description:Displacement of [3H]GR-113808 from 5HT4 receptor in guinea pig striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50092558(4-Amino-5-chloro-2-methoxy-benzoic acid 2-[4-(2-ch...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4E receptor isoform expressed in C6 glial cells incubated with 0.2 nM [3H]-GR-113,...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50174443(1-[2-(4-amino-5-chloro-2-methoxyphenylcarbonyloxy)...)
Affinity DataKi:  10nMAssay Description:Binding affinity for 5-HT4 receptor using [3H]-GR-113,808More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM29526(2-Piperidinoethyl 4-amino-5-chloro-2-methoxybenzoa...)
Affinity DataKi:  10.7nMAssay Description:Binding affinity was determined against cloned 5-hydroxytryptamine 4B receptor isoform expressed in COS-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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