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TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 50nMAssay Description:Inhibition of Electrophorus electricus C2888 AChE using acetylthiocholine iodide as substrate by Ellman's spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50012188(6BIO)
Affinity DataIC50: 52nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 74nMAssay Description:Inhibition of Electrophorus electricus AChE after 120 secs by Ellman spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 75nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 80nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 5(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50012188(6BIO)
Affinity DataIC50: 85nMAssay Description:Inhibition of CDK5 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Rat)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 90nMAssay Description:Inhibition of rat DYRK1A assessed as inhibition of phosphate incorporation using GRSRSRSRSRSR and [gamma-33P]ATP as substrate after 30 mins by scinti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 160nMAssay Description:Inhibition of electric eel AChE preincubated for 15 mins followed by addition of acetylthiocholine iodide as substrate measured after 30 mins by Ellm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 170nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Mouse)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 210nMAssay Description:Inhibition of mouse recombinant GST-fused CLK1 expressed in Escherichia coli cells assessed as inhibition of phosphate incorporation using GRSRSRSRSR...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK4(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 220nMAssay Description:Inhibition of CLK4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 220nMAssay Description:Inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50012188(6BIO)
Affinity DataIC50: 320nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 350nMAssay Description:Inhibition of DYRK1B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50004000(CHEMBL94 | physostigmine | Antilirium | Eserine | ...)
Affinity DataIC50: 580nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine chloride as substrate measured after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK2(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 680nMAssay Description:Inhibition of CLK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50330755(Mesuagenin B | CHEMBL1277588)
Affinity DataIC50: 700nMAssay Description:Inhibition of Electrophorus electricus AChE after 120 secs by Ellman spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 820nMAssay Description:Inhibition of CDK9/cyclin T (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 1.03E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50330754(Mesuagenin A | CHEMBL1277495)
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of Electrophorus electricus AChE after 120 secs by Ellman spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 3(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of DYRK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182487(Malabaricone A)
Affinity DataIC50: 1.31E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355395(CHEMBL1834806)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355396(CHEMBL1834808)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355395(CHEMBL1834806)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of DYRK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182486(MALABARICONE B)
Affinity DataIC50: 1.76E+3nMAssay Description:Inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355396(CHEMBL1834808)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182486(MALABARICONE B)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182491(CHEBI:69015 | Malabaricone C)
Affinity DataIC50: 1.94E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355397(CHEMBL1834807)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK1(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50012188(6BIO)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of CLK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355398(CHEMBL1834809)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021613(Atolaphyllidine)
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetDual specificity protein kinase CLK3(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of CLK3 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355397(CHEMBL1834807)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182491(CHEBI:69015 | Malabaricone C)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of equine serum BChE using S-butyrylthiocholine chloride as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50330760(5,7-dihydroxy-8-(3-methylbutanoyl)-6-[(E)-3,7-dime...)
Affinity DataIC50: 3.06E+3nMAssay Description:Inhibition of Electrophorus electricus AChE after 120 secs by Ellman spectroscopic methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355398(CHEMBL1834809)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355399(CHEMBL1834877)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCholinesterase(Horse)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50187684(CHEMBL3827910)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of equine serum BChE preincubated for 15 mins followed by addition of S-butyrylthiocholine chloride as substrate measured after 30 mins by...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/8/2017
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355399(CHEMBL1834877)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355400(CHEMBL1834810)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021616(CHEMBL3297832)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of CDK1 (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Electric eel)
Guangzhou University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50355401(CHEMBL1834811)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibition of electric eel AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Institut De Chimie Des Substances Naturelles

Curated by ChEMBL
LigandPNGBDBM50021614(CHEMBL3297831)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of DYRK1A (unknown origin) assessed as inhibition of phosphate incorporation into substrate in presence of radiolabeled ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355400(CHEMBL1834810)
Affinity DataIC50: 5.90E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50355401(CHEMBL1834811)
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of human recombinant AChE using acetylthiocholine iodide as substrate by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/24/2012
Entry Details Article
PubMed
TargetAcetylcholinesterase(Human)
University of Malaya

Curated by ChEMBL
LigandPNGBDBM50182488(CHEMBL3819036)
Affinity DataIC50: 6.44E+3nMAssay Description:Inhibition of AChE (unknown origin) using acetylthiocholine iodide as substrate incubated for 30 mins by Ellman's microplate assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2017
Entry Details Article
PubMed
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