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TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333703(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333704(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333705(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333706(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333707(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333708(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333711(N-tert-butyl-2-(2-tert-butyl-1-(2-(tert-butylamino...)
Affinity DataEC50:  570nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333713(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxo-1-(py...)
Affinity DataEC50:  600nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333716(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50:  740nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333719(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50:  940nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333722(N-tert-butyl-2-(1-(2-(tert-butylamino)-2-oxoethyl)...)
Affinity DataEC50:  1.81E+3nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333723(N-tert-butyl-5-(1-(tert-butylamino)-2-methyl-1-oxo...)
Affinity DataEC50:  6.64E+3nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50333724(2-(2-(3,5-bis(trifluoromethyl)phenyl)-1-(2-(tert-b...)
Affinity DataEC50:  1.08E+4nMAssay Description:Activity at PXR by induction assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394606(CHEMBL2164226)
Affinity DataEC50:  99nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50:  130nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394607(CHEMBL2164225)
Affinity DataEC50:  95nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394608(CHEMBL2164224)
Affinity DataEC50:  147nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394606(CHEMBL2164226)
Affinity DataEC50:  1.00E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50381914(MK-7725 | CHEMBL2023109)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394607(CHEMBL2164225)
Affinity DataEC50: >3.00E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394608(CHEMBL2164224)
Affinity DataEC50:  2.40E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394609(CHEMBL2164223)
Affinity DataEC50:  83nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394610(CHEMBL2164222)
Affinity DataEC50:  134nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394611(CHEMBL2164582)
Affinity DataEC50:  89nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394612(CHEMBL2164581)
Affinity DataEC50:  93nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394613(CHEMBL2164580)
Affinity DataEC50:  57nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394614(CHEMBL2164579)
Affinity DataEC50:  76nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394615(CHEMBL2164578)
Affinity DataEC50:  115nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394616(CHEMBL2164577)
Affinity DataEC50:  102nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataEC50:  58nMAssay Description:Agonist activity at mouse BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394609(CHEMBL2164223)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394610(CHEMBL2164222)
Affinity DataEC50:  69nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394611(CHEMBL2164582)
Affinity DataEC50:  52nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394612(CHEMBL2164581)
Affinity DataEC50:  56nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394613(CHEMBL2164580)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394614(CHEMBL2164579)
Affinity DataEC50:  77nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394615(CHEMBL2164578)
Affinity DataEC50:  114nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394616(CHEMBL2164577)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBombesin receptor subtype-3(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataEC50:  42nMAssay Description:Agonist activity at human BRS-3 expressed in HEK293AEQ cells assessed as bioluminescence for 10 mins by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394609(CHEMBL2164223)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394610(CHEMBL2164222)
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394611(CHEMBL2164582)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394612(CHEMBL2164581)
Affinity DataEC50:  3.50E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394613(CHEMBL2164580)
Affinity DataEC50:  1.18E+4nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394614(CHEMBL2164579)
Affinity DataEC50:  1.90E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394615(CHEMBL2164578)
Affinity DataEC50:  6.60E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394616(CHEMBL2164577)
Affinity DataEC50:  1.10E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394617(CHEMBL2164576)
Affinity DataEC50:  1.80E+3nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetNuclear receptor subfamily 1 group I member 2(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50394618(CHEMBL2164575)
Affinity DataEC50:  677nMAssay Description:Activation of PXRMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50434313(CHEMBL2386571)
Affinity DataKd:  0.800nMAssay Description:Binding affinity to FAAH in human cortical homogenatesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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