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TargetD(2) dopamine receptor(Rat)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataKd:  0.0400nMAssay Description:Binding affinity against Dopamine receptor D2 in rat striatum using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor beta using rabbit saphenous vein assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetD(1A) dopamine receptor(Rat)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataKd:  0.300nMAssay Description:Binding affinity against dopamine receptor D1 in rat striatum using [3H]SCH-23390 as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataKd:  1.80nMAssay Description:Binding affinity against 5-hydroxytryptamine 1 receptor using rabbit jugular vein assay in the absence of endotheliumMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataKd:  1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor beta using rabbit saphenous vein assay.More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005835(Sumax | 3-[2-(dimethylamino)ethyl]-N-methylindole-...)
Affinity DataIC50: 0.501nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataIC50: 2.80nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50005835(Sumax | 3-[2-(dimethylamino)ethyl]-N-methylindole-...)
Affinity DataIC50: 3nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473516(CHEMBL2110299)
Affinity DataIC50: 3.60nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50033383((S)-4-((3-(2-(dimethylamino)ethyl)-1H-indol-5-yl)m...)
Affinity DataIC50: 6.20nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473505(CHEMBL2368256)
Affinity DataIC50: 7.10nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473521(CP-122288 | CHEMBL159332)
Affinity DataIC50: 7.20nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473512(CHEMBL2368254)
Affinity DataIC50: 9.5nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473512(CHEMBL2368254)
Affinity DataIC50: 14nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473521(CP-122288 | CHEMBL159332)
Affinity DataIC50: 14nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473508(CHEMBL158638)
Affinity DataIC50: 15nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 15.8nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473516(CHEMBL2110299)
Affinity DataIC50: 18nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473504(CHEMBL3084967)
Affinity DataIC50: 29nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473505(CHEMBL2368256)
Affinity DataIC50: 32nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017914(CHEMBL353950 | 3-(1-Ethyl-5-pyridin-3-ylmethyl-1H-...)
Affinity DataIC50: 42nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017903(CHEMBL170754 | 3-(1-tert-Butyl-5-pyridin-3-ylmethy...)
Affinity DataIC50: 44nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473508(CHEMBL158638)
Affinity DataIC50: 45nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50017905(CHEMBL352763 | 2-Methyl-3-(1-methyl-5-pyridin-3-yl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of thromboxane A2 synthetase as reduced ADP-induced aggregation of human platelet rich plasma in the presence of pig aortal microsomesMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473509(CHEMBL2368257)
Affinity DataIC50: 57.5nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473509(CHEMBL2368257)
Affinity DataIC50: 58nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473501(CHEMBL2368253)
Affinity DataIC50: 65nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000334(Agrylin | 6,7-Dichloro-1,5-dihydro-imidazo[2,1-b]q...)
Affinity DataIC50: 82nMAssay Description:Inhibition of human blood platelet c-AMP phosphodiesteraseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 89nMAssay Description:Binding affinity against calf caudate 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473509(CHEMBL2368257)
Affinity DataIC50: 97.7nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473501(CHEMBL2368253)
Affinity DataIC50: 98nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473509(CHEMBL2368257)
Affinity DataIC50: 98nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 100nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 100nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 112nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473502(CHEMBL159470)
Affinity DataIC50: 141nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473504(CHEMBL3084967)
Affinity DataIC50: 141nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 162nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 162nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473520(CHEMBL2368259)
Affinity DataIC50: 191nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473510(CHEMBL2368261)
Affinity DataIC50: 195nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473510(CHEMBL2368261)
Affinity DataIC50: 204nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473513(CHEMBL350277)
Affinity DataIC50: 263nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473520(CHEMBL2368259)
Affinity DataIC50: 275nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1B(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473502(CHEMBL159470)
Affinity DataIC50: 316nMAssay Description:Binding affinity in CHO-K1 cells transfected with human recombinant 5-hydroxytryptamine 1B receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473513(CHEMBL350277)
Affinity DataIC50: 339nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000308(CHEMBL158201 | 6-(Imidazol-1-yl-phenyl-methyl)-3,4...)
Affinity DataIC50: 350nMAssay Description:Compound was evaluated for the inhibition of human blood platelet,thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1F(Human)
Glaxowellcome

Curated by ChEMBL
LigandPNGBDBM50473503(CHEMBL2110300)
Affinity DataIC50: 363nMAssay Description:Binding affinity towards human recombinant 5-hydroxytryptamine 1F receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetThromboxane-A synthase(Human)
Syntex Research

Curated by ChEMBL
LigandPNGBDBM50000318(CHEMBL347379 | 6-(2-Imidazol-1-yl-vinyl)-1H-quinol...)
Affinity DataIC50: 380nMAssay Description:Compound was evaluated for the inhibition of human blood platelet,thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target5-hydroxytryptamine receptor 1D(Human)
Wellcome Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50473515(CHEMBL2368255)
Affinity DataIC50: 501nMAssay Description:Binding affinity in CHO-K1 cells transfected with human 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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