Compile Data Set for Download or QSAR
Report error Found 286 with Last Name = 'mazza' and Initial = 'f'
TargetStromelysin-1(Human)
Istituto Di Cristallografia

LigandPNGBDBM12073((S)-[1-(4-Methoxybiphenyl-4-sulfonylamino)-2-methy...)
Affinity DatapH: 7.5 T: 2°CAssay Description:Inhibition of the matrix metalloproteinases MMP-2, MMP-3, and MMP-8 has been determined by continuously monitoring the hydrolysis of the fluorescent ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2006
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28759(CHEMBL191275 | (2S)-3-phenyl-2-(4-phenylphenoxy)pr...)
Affinity DataEC50:  480nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28760((2R)-3-phenyl-2-(4-phenylphenoxy)propanoic acid | ...)
Affinity DataEC50:  5.93E+3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  40nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28759(CHEMBL191275 | (2S)-3-phenyl-2-(4-phenylphenoxy)pr...)
Affinity DataEC50:  220nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  1.62E+3nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28759(CHEMBL191275 | (2S)-3-phenyl-2-(4-phenylphenoxy)pr...)
Affinity DataEC50:  260nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  40nMAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28760((2R)-3-phenyl-2-(4-phenylphenoxy)propanoic acid | ...)
Affinity DataAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28760((2R)-3-phenyl-2-(4-phenylphenoxy)propanoic acid | ...)
Affinity DataAssay Description:The HepG2 cells were co-transfected with DNA construct containing PPAR-Gal4 chimeric receptor and Gal4-luciferase reporter. The luciferase activity w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataKd:  14.8nM EC50:  3.80nMpH: 7.5 T: 2°CAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28762((2R)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKd:  685nM EC50:  73.3nMpH: 7.5 T: 2°CAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28763((2S)-2-(4-{2-[1,3-benzoxazol-2-yl(heptyl)amino]eth...)
Affinity DataKd:  1.98E+3nM EC50:  593nMpH: 7.5 T: 2°CAssay Description:Kd values were obtained by incubating His-PPARgamma-LBD with biotinylated peptide, europium-labeled anti-histidine antibody, and allophycocyanin-labe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/7/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299112((S)-2-(4-phenethylphenoxy)-3-phenylpropanoic acid ...)
Affinity DataEC50:  860nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299109((S)-2-(4-benzylphenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  580nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299109((S)-2-(4-benzylphenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299112((S)-2-(4-phenethylphenoxy)-3-phenylpropanoic acid ...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299109((S)-2-(4-benzylphenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28681(cid_5281055 | [3H]rosiglitazone | CHEMBL121 | ROSI...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299110(rac-2-(4-Phenoxy-phenoxy)-3-phenyl-propanoic Acid ...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299111(rac-2-(4-Benzyloxy-phenoxy)-3-phenyl-propanoic Aci...)
Affinity DataEC50:  107nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299113(rac-2-(4-cis-Styryl-phenoxy)-3-phenyl-propanoic Ac...)
Affinity DataEC50:  160nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28759(CHEMBL191275 | (2S)-3-phenyl-2-(4-phenylphenoxy)pr...)
Affinity DataEC50:  190nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299114(rac-2-(4-Phenylthiomethyl-phenoxy)-3-phenyl-propan...)
Affinity DataEC50:  310nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299112((S)-2-(4-phenethylphenoxy)-3-phenylpropanoic acid ...)
Affinity DataEC50:  330nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299112((S)-2-(4-phenethylphenoxy)-3-phenylpropanoic acid ...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299114(rac-2-(4-Phenylthiomethyl-phenoxy)-3-phenyl-propan...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299115(rac-2-(4-Benzylthio-phenoxy)-3-phenyl-propanoic Ac...)
Affinity DataEC50:  488nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299116(rac-2-(4-Phenylethynyl-phenoxy)-3-phenyl-propanoic...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM28759(CHEMBL191275 | (2S)-3-phenyl-2-(4-phenylphenoxy)pr...)
Affinity DataEC50:  560nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299109((S)-2-(4-benzylphenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  572nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299117(rac-2-(4-Phenoxymethyl-phenoxy)-3-phenyl-propanoic...)
Affinity DataEC50:  600nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299118(rac-2-(4-trans-Styryl-phenoxy)-3-phenyl-propanoic ...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299119(rac-2-[4-(3-Phenyl-propyl)phenoxy]-3-phenyl-propan...)
Affinity DataEC50:  720nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299119(rac-2-[4-(3-Phenyl-propyl)phenoxy]-3-phenyl-propan...)
Affinity DataEC50:  870nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299110(rac-2-(4-Phenoxy-phenoxy)-3-phenyl-propanoic Acid ...)
Affinity DataEC50:  1.21E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299116(rac-2-(4-Phenylethynyl-phenoxy)-3-phenyl-propanoic...)
Affinity DataEC50:  1.36E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299115(rac-2-(4-Benzylthio-phenoxy)-3-phenyl-propanoic Ac...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299120(rac-2-(4-Phenylaminomethyl-phenoxy)-3-phenyl-propa...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299113(rac-2-(4-cis-Styryl-phenoxy)-3-phenyl-propanoic Ac...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299121((R)-2-(4-Phenethyl-phenoxy)-3-phenyl-propanoic Aci...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM24566(JMC515449 Compound 1 | Wyeth 14,643 | 2-({4-chloro...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299118(rac-2-(4-trans-Styryl-phenoxy)-3-phenyl-propanoic ...)
Affinity DataEC50:  1.75E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299122(rac-2-(4-Phenylacetyl-phenoxy)-3-phenyl-propanoic ...)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299123((R)-2-(4-Benzyl-phenoxy)-3-phenyl-propanoic Acid |...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299111(rac-2-(4-Benzyloxy-phenoxy)-3-phenyl-propanoic Aci...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299117(rac-2-(4-Phenoxymethyl-phenoxy)-3-phenyl-propanoic...)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299124(rac-2-(4-Benzylamino-phenoxy)-3-phenyl-propanoic A...)
Affinity DataEC50:  3.60E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299123((R)-2-(4-Benzyl-phenoxy)-3-phenyl-propanoic Acid |...)
Affinity DataEC50:  5.70E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Consiglio Nazionale Delle Ricerche

LigandPNGBDBM50299122(rac-2-(4-Phenylacetyl-phenoxy)-3-phenyl-propanoic ...)
Affinity DataEC50:  9.10E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in human HepG2 cells assessed as receptor transactivation by lucifera...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2010
Entry Details Article
PubMed
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