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TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521644(CHEMBL4592246)
Affinity DataKd:  9.80E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521645(CHEMBL4575624)
Affinity DataKd:  490nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521646(CHEMBL4520983)
Affinity DataKd:  570nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521647(CHEMBL4447862)
Affinity DataKd:  1.49E+4nMAssay Description:Binding affinity to BRAF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521648(CHEMBL4579756)
Affinity DataKd:  2.96E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521649(CHEMBL4531640)
Affinity DataKd:  3.89E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521650(CHEMBL4441432)
Affinity DataKd:  1.09E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521651(CHEMBL4440248)
Affinity DataKd:  2.20E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521652(CHEMBL4459130)
Affinity DataKd:  4.75E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521653(CHEMBL4589790)
Affinity DataKd:  1.88E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521654(CHEMBL4541462)
Affinity DataKd:  130nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521655(CHEMBL4520561)
Affinity DataKd:  480nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521656(CHEMBL4458911)
Affinity DataKd:  450nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521657(CHEMBL4471635)
Affinity DataKd:  360nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521658(CHEMBL4542330)
Affinity DataKd:  2.69E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521659(CHEMBL4447430)
Affinity DataKd:  540nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521660(CHEMBL4446282)
Affinity DataKd:  190nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521661(CHEMBL4457586)
Affinity DataKd:  780nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521662(CHEMBL4471788)
Affinity DataKd:  460nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521663(CHEMBL4443180)
Affinity DataKd:  61nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521654(CHEMBL4541462)
Affinity DataKd:  350nMAssay Description:Binding affinity to BRAF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521664(CHEMBL4541688)
Affinity DataKd:  3.84E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521665(CHEMBL4542044)
Affinity DataKd:  540nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521666(CHEMBL4443036)
Affinity DataKd:  1.25E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521667(CHEMBL4474883)
Affinity DataKd:  800nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521668(CHEMBL4450992)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521669(CHEMBL4463173)
Affinity DataKd:  360nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521670(CHEMBL4546018)
Affinity DataKd:  1.89E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521671(CHEMBL4448348)
Affinity DataKd:  1.02E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521647(CHEMBL4447862)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521672(CHEMBL4444440)
Affinity DataKd:  5.75E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521673(CHEMBL4441999)
Affinity DataKd:  550nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521674(CHEMBL4561891)
Affinity DataKd:  4.10E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521662(CHEMBL4471788)
Affinity DataKd:  310nMAssay Description:Binding affinity to BRAF (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase B-raf(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50521675(CHEMBL4547059)
Affinity DataKd:  2.40E+3nMAssay Description:Binding affinity to BRAF (unknown origin) by intrinsic tryptophan fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50582005(CHEMBL5093856)
Affinity DataEC50:  650nMAssay Description:Binding affinity to PLK1 in human PC-3 cells incubated for 2 hrs followed by heat shock for 10 mins by cellular thermal shift assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase haspin(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity to human HASPIN assessed as dissociation constant by KdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMitogen-activated protein kinase kinase kinase kinase 2(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  940nMAssay Description:Binding affinity to human MAP4K2 assessed as dissociation constant by KdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetMyosin-IIIb(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd: >3.00E+4nMAssay Description:Binding affinity to human MYO3B assessed as dissociation constant by KdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-C(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50248629(CHEMBL4076837 | US11471446, Compound DBA-9)
Affinity DataKd:  2nMAssay Description:Binding affinity to kinase tracer 236 binding to His tagged recombinant human CDK8/cyclinC assessed as dissociation constant by TR FRET based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-C(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  1.40nMAssay Description:Binding affinity to kinase tracer 236 binding to His tagged recombinant human CDK8/cyclinC assessed as dissociation constant by TR FRET based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50248629(CHEMBL4076837 | US11471446, Compound DBA-9)
Affinity DataKd:  3nMAssay Description:Binding affinity to recombinant human CDK19/cyclinC assessed as dissociation constant by TR FRET based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-C/Cyclin-dependent kinase 19(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  2.90nMAssay Description:Binding affinity to recombinant human CDK19/cyclinC assessed as dissociation constant by TR FRET based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 8(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  55nMAssay Description:Binding affinity to human CDK8 assessed as dissociation constant by KdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 19(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataKd:  44nMAssay Description:Binding affinity to human CDK19 assessed as dissociation constant by KdELECT Discover assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50596070(CHEMBL5180726)
Affinity DataEC50:  820nMAssay Description:Binding affinity to full length PLK1 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 56...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50596070(CHEMBL5180726)
Affinity DataEC50:  6.90E+3nMAssay Description:Binding affinity to full length PLK3 in human PC-3 cells assessed as stabilized protein incubated for 2 hrs followed by aggregation temperature at 48...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
PubMed
TargetCyclin-A2(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50059785(CHEMBL3393766)
Affinity DataKd:  19nMAssay Description:Binding affinity to cyclin A2 (174 to 432) (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Human)
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50117496(H-His-Ala-Lys-Arg-Arg-Leu-Ile-(L)-Pse-OH | CHEMBL4...)
Affinity DataIC50: 2nMAssay Description:In vitro inhibition of CDK2-cyclin A kinase activity on retinoblastoma proteinMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-C(Human)
University of South Carolina

Curated by ChEMBL
LigandPNGBDBM50585694(CHEMBL4878072)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of kinase tracer 236 binding to His tagged recombinant human CDK8/cyclin C incubated for 60 min FRET based LanthaScreen Eu-Kinase binding ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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