Compile Data Set for Download or QSAR
Report error Found 553 with Last Name = 'miguel' and Initial = 'ts'
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392770(CHEMBL2151243)
Affinity DataIC50: 0.990nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383838(CHEMBL2030996)
Affinity DataIC50: 1nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383838(CHEMBL2030996)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392782(CHEMBL2151237)
Affinity DataIC50: 2nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392785(CHEMBL2151240)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392770(CHEMBL2151243)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392780(CHEMBL2151235)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392782(CHEMBL2151237)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392786(CHEMBL2151241)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392776(CHEMBL2151151)
Affinity DataIC50: 3.10nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392771(CHEMBL2151244)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392773(CHEMBL2151148)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392777(CHEMBL2151152)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392783(CHEMBL2151238)
Affinity DataIC50: 4nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392780(CHEMBL2151235)
Affinity DataIC50: 4nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392786(CHEMBL2151241)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392787(CHEMBL2151242)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392783(CHEMBL2151238)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383839(CHEMBL2030997)
Affinity DataIC50: 5nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392777(CHEMBL2151152)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392776(CHEMBL2151151)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392781(CHEMBL2151236)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383837(CHEMBL2030998)
Affinity DataIC50: 6.60nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383837(CHEMBL2030998)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50394892(CHEMBL2165051)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant GST-tagged mTOR-mediated 4EBP1 phosphorylation after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50432336(CHEMBL2348154)
Affinity DataIC50: 7nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392775(CHEMBL2151150)
Affinity DataIC50: 7.20nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392787(CHEMBL2151242)
Affinity DataIC50: 7.60nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50341063(2-(4-(2-(3-hydroxyphenylamino)-1H-benzo[d]imidazol...)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant GST-tagged mTOR-mediated 4EBP1 phosphorylation after 90 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392778(CHEMBL2151153)
Affinity DataIC50: 8.30nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392771(CHEMBL2151244)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392773(CHEMBL2151148)
Affinity DataIC50: 8.80nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50432334(CHEMBL2348153)
Affinity DataIC50: 9nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392784(CHEMBL2151239)
Affinity DataIC50: 11nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50432343(CHEMBL2348156)
Affinity DataIC50: 11nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50383839(CHEMBL2030997)
Affinity DataIC50: 12nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392778(CHEMBL2151153)
Affinity DataIC50: 13nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392779(CHEMBL2151154)
Affinity DataIC50: 14nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392784(CHEMBL2151239)
Affinity DataIC50: 18nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392781(CHEMBL2151236)
Affinity DataIC50: 18nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50432365(CHEMBL2348182)
Affinity DataIC50: 25nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392785(CHEMBL2151240)
Affinity DataIC50: 26nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50394846(CHEMBL2165017 | US8772480, 35)
Affinity DataIC50: 29nMAssay Description:Inhibition of PIK3C2betaMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50432335(CHEMBL2348152)
Affinity DataIC50: 30nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50401254(CHEMBL2206906 | US8772480, 335)
Affinity DataIC50: 32nMAssay Description:Inhibition of recombinant N-terminal GST-tagged mTOR using GFP-4EBP as substrate after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392772(CHEMBL2151316)
Affinity DataIC50: 44nMAssay Description:Inhibition of BACEMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCyclin-dependent kinase 2(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50432341(CHEMBL2348155)
Affinity DataIC50: 60nMAssay Description:Inhibition of CDK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetBeta-secretase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50392779(CHEMBL2151154)
Affinity DataIC50: 65nMAssay Description:Inhibition of BACE by cells based assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50429636(CHEMBL2334964 | US9616064, Compound 15d)
Affinity DataIC50: 66nMAssay Description:Inhibition of CDC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSerine/threonine-protein kinase mTOR(Human)
Amgen

Curated by ChEMBL
LigandPNGBDBM50401256(CHEMBL2206904 | US8772480, 331)
Affinity DataIC50: 74nMAssay Description:Inhibition of recombinant N-terminal GST-tagged mTOR using GFP-4EBP as substrate after 90 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Displayed 1 to 50 (of 553 total ) | Next | Last >>
Jump to: