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TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296336((3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl...)
Affinity DataKi:  0.0600nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank


TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296336((3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl...)
Affinity DataKi:  0.0700nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296329((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phe...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296329((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phe...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296329((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phe...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296336((3R)-3-{[(2S)-2-Cyclopentyl-2-hydroxy-2-(2-thienyl...)
Affinity DataKi:  0.0900nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)
Affinity DataKi:  0.100nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)
Affinity DataKi:  0.120nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50296345((1R,2R,4S,5R,7S)-7-(2-hydroxy-2,2-di-thiophen-2-yl...)
Affinity DataKi:  0.140nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336996(CHEMBL1672631 | N-[6-(2-Fluorophenyl)-5-(3-fluorop...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M3(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50378083(Atrovent HFA | IPRATROPIUM BROMIDE)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to muscarinic M3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336991(CHEMBL1672623 | N-[6-(2-Fluorophenyl)-5-pyridin-4-...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M2(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50378083(Atrovent HFA | IPRATROPIUM BROMIDE)
Affinity DataKi:  1.02nMAssay Description:Binding affinity to muscarinic M2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336989(CHEMBL1672619 | N-[6-(5-Methyl-2-furyl)-5-pyridin-...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMuscarinic acetylcholine receptor M1(Human)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50378083(Atrovent HFA | IPRATROPIUM BROMIDE)
Affinity DataKi:  1.51nMAssay Description:Binding affinity to muscarinic M1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336980(CHEMBL1672633 | N-[5-(3-Fluoropyridin-4-yl)-6-(1,3...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336989(CHEMBL1672619 | N-[6-(5-Methyl-2-furyl)-5-pyridin-...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336974(CHEMBL1672611 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336985(CHEMBL1672615 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336983(CHEMBL1672613 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336982(CHEMBL1672612 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336979(CHEMBL1672632 | N-[5-(3-Fluoropyridin-4-yl)-6-(1,3...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336984(CHEMBL1672614 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336978(CHEMBL1672630 | N-(5-(3-chloropyridin-4-yl)-6-(pyr...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336990(CHEMBL1672620 | N-(6-Pyridin-2-yl-5-pyridin-4-ylpy...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336989(CHEMBL1672619 | N-[6-(5-Methyl-2-furyl)-5-pyridin-...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336988(2-Cyclopentyl-N-[6-(2-furyl)-5-pyridin-4-ylpyrazin...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336986(CHEMBL1672616 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336985(CHEMBL1672615 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336984(CHEMBL1672614 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336977(CHEMBL1672627 | N-[5-(3-Fluoropyridin-4-yl)-6-pyri...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336975(CHEMBL1672621 | N-(6-Pyridin-3-yl-5-pyridin-4-ylpy...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336991(CHEMBL1672623 | N-[6-(2-Fluorophenyl)-5-pyridin-4-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336981(CHEMBL1672629 | N-[5-(3,5-Difluoropyridin-4-yl)-6-...)
Affinity DataKi:  26nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336986(CHEMBL1672616 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336994(CHEMBL1672626 | N-[6-(2-Furyl)-5-pyrimidin-4-ylpyr...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336976(CHEMBL1672622 | N-(5,6-Dipyridin-4-ylpyrazin-2-yl)...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336983(CHEMBL1672613 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336993(CHEMBL1672625 | N-[6-(1,3-Oxazol-5-yl)-5-pyridin-4...)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336974(CHEMBL1672611 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336991(CHEMBL1672623 | N-[6-(2-Fluorophenyl)-5-pyridin-4-...)
Affinity DataKi:  51nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2a(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336983(CHEMBL1672613 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336974(CHEMBL1672611 | N-[6-(2-Furyl)-5-pyridin-4-ylpyraz...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336992(CHEMBL1672624 | N-(6-(oxazol-2-yl)-5-(pyridin-4-yl...)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336987(4-Fluoro-N-[6-(2-furyl)-5-pyridin-4-ylpyrazin-2-yl...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A2b(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336995(CHEMBL1672628 | N-[5-(3-Chloropyridin-4-yl)-6-pyri...)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]DPCPX from human adenosine A2B receptor expressed in HEK293 cells after 60 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetAdenosine receptor A1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50336988(2-Cyclopentyl-N-[6-(2-furyl)-5-pyridin-4-ylpyrazin...)
Affinity DataKi:  98nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cells after 90 mins by filtration binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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