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TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401097(CHEMBL2204469)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity to human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401116(CHEMBL2204474)
Affinity DataIC50: 0.800nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006915(CHEMBL3236929)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006823(CHEMBL3236950)
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401097(CHEMBL2204469)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of CRTH2 receptor-mediated chemotaxis in human basophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006830(CHEMBL3236948)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of CRTH2 receptor-mediated chemotaxis in human basophilsMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006830(CHEMBL3236948)
Affinity DataIC50: 1.40nMAssay Description:Binding affinity to human CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401108(CHEMBL2205148)
Affinity DataIC50: 2nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006891(CHEMBL3236958)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401097(CHEMBL2204469)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401097(CHEMBL2204469)
Affinity DataIC50: 3nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006818(CHEMBL3236951)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006823(CHEMBL3236950)
Affinity DataIC50: 3nMT: 2°CAssay Description:Antagonist activity at CRTh2 in human peripheral blood assessed as inhibition of PGD2-induced eosinophil shape change at room temperature by flow cyt...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006894(CHEMBL3236955)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006899(CHEMBL3237239)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401120(CHEMBL2204470)
Affinity DataIC50: 4nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006827(CHEMBL3236949)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006830(CHEMBL3236948)
Affinity DataIC50: 4nMAssay Description:Inhibition of mouse CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006880(CHEMBL3236960)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006896(CHEMBL3237242)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401118(CHEMBL2204472)
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006870(CHEMBL3237230)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006893(CHEMBL3236956)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401117(CHEMBL2204473)
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006830(CHEMBL3236948)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006865(CHEMBL3237233)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006866(CHEMBL3237232)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006895(CHEMBL3237243)
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401111(CHEMBL2204479)
Affinity DataIC50: 7nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Mouse)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401097(CHEMBL2204469)
Affinity DataIC50: 7nMAssay Description:Inhibition of mouse CRTH2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006892(CHEMBL3236957)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006830(CHEMBL3236948)
Affinity DataIC50: 8nMT: 2°CAssay Description:Antagonist activity at CRTh2 in human peripheral blood assessed as inhibition of PGD2-induced eosinophil shape change at room temperature by flow cyt...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006890(CHEMBL3236959)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006897(CHEMBL3237241)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006898(CHEMBL3237240)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006918(CHEMBL3236945)
Affinity DataIC50: 8nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401122(CHEMBL2205146)
Affinity DataIC50: 9nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401119(CHEMBL2204471)
Affinity DataIC50: 10nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401122(CHEMBL2205146)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006920(CHEMBL3236943)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401124(CHEMBL2205144)
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401126(CHEMBL2204493)
Affinity DataIC50: 11nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006873(CHEMBL3237228)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006900(CHEMBL3237238)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401113(CHEMBL2204477)
Affinity DataIC50: 12nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50006802(CHEMBL3236952)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human recombinant CRTh2 expressed in CHO-K1 cells by cAMP TR FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401115(CHEMBL2204475)
Affinity DataIC50: 15nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401106(CHEMBL2205150)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401112(CHEMBL2204478)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProstaglandin D2 receptor 2(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50401121(CHEMBL2205147)
Affinity DataIC50: 16nMAssay Description:Displacement of [3H]PGD2 from recombinant human CRTH2 receptor expressed in CHO-K1 cells after 30 min by FRET methodMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
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