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TargetMelanin-concentrating hormone receptor 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295693(CHEMBL557629)
Affinity DataKi:  0.0340nMAssay Description:Displacement of [35S] 4-(1-(3,4-difluorophenyl)-2-(ethyl(3-(6-fluoro-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)amino)-2-oxoethyl)-3-oxopip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295693(CHEMBL557629)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [35S] 4-(1-(3,4-difluorophenyl)-2-(ethyl(3-(6-fluoro-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)amino)-2-oxoethyl)-3-oxopip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.170nMAssay Description:Inhibition of [3H]PDBu binding to PKCbeta C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Rat)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50000066((2-Azepan-1-yl-ethyl)-[2-(3,4-dichloro-phenyl)-eth...)
Affinity DataKi:  0.170nMAssay Description:Inhibition of [3H]-NANM binding to sigma receptor obtained from tissue homogenate preparation of fresh whole rat brain minus cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.180nMAssay Description:Displacement of [3H]PDBu from PKCeta C1B domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295690((+/-)-2-(3,4-difluorophenyl)-N-ethyl-N-(3-(6-fluor...)
Affinity DataKi:  0.180nMAssay Description:Binding affinity to human MCH1R expressed in CHO cells by scintillation counting per mg of proteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]PDBu from PKCtheta C1B domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1A receptor in rat submaxillary gland membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.260nMAssay Description:Inhibition of [3H]PDBu binding to PKCalpha C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]PDBu from PKCdelta C1B domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295690((+/-)-2-(3,4-difluorophenyl)-N-ethyl-N-(3-(6-fluor...)
Affinity DataKi:  0.420nMAssay Description:Displacement of [35S] 4-(1-(3,4-difluorophenyl)-2-(ethyl(3-(6-fluoro-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)amino)-2-oxoethyl)-3-oxopip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C eta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.450nMAssay Description:Inhibition of [3H]PDBu binding to PKCeta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.460nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mouse)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295690((+/-)-2-(3,4-difluorophenyl)-N-ethyl-N-(3-(6-fluor...)
Affinity DataKi:  0.5nMAssay Description:Displacement of [35S] 4-(1-(3,4-difluorophenyl)-2-(ethyl(3-(6-fluoro-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)amino)-2-oxoethyl)-3-oxopip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  0.540nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50343939((S)-2-(6-hydroxy-6-methylheptan-2-ylamino)-4-methy...)
Affinity DataKi:  0.590nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115122(CHEMBL3609360)
Affinity DataKi:  0.610nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187753(6-fluoro-3-(1-(3-(piperidin-1-yl)propyl)piperidin-...)
Affinity DataKi:  0.630nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)
Affinity DataKi:  0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C gamma type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50343939((S)-2-(6-hydroxy-6-methylheptan-2-ylamino)-4-methy...)
Affinity DataKi: <1nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]PDBu from PKCalpha C1A domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206860(CHEMBL3974799)
Affinity DataKi:  1nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206864(CHEMBL3903916)
Affinity DataKi: <1nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434226(CHEMBL2385483)
Affinity DataKi:  1nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187752(3-(1-(4-(piperidin-1-yl)butyl)piperidin-4-yl)-1H-i...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50343938(CHEMBL1778662 | rac-2-(6-hydroxy-6-methylheptan-2-...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]PDBu from PKCepsilon C1B domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187747(3-(1-(5-(piperidin-1-yl)pentyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C beta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]PDBu from PKCbeta C1A domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 2(Human)
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50295693(CHEMBL557629)
Affinity DataKi:  1.60nMAssay Description:Displacement of [35S] 4-(1-(3,4-difluorophenyl)-2-(ethyl(3-(6-fluoro-3H-spiro[isobenzofuran-1,4'-piperidine]-1'-yl)propyl)amino)-2-oxoethyl)-3-oxopip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM13534(CHEMBL572878 | N-[4-({4-[(3-methyl-1H-pyrazol-5-yl...)
Affinity DataKi:  2nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50004205(MK-045 | MK-0457 | TOZASERTIB | US9249124, VX680 |...)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMacrophage metalloelastase(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50294120(2-(biphenyl-4-ylsulfonamido)-N-hydroxyacetamide | ...)
Affinity DataKi:  2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Human)
University of Florence

Curated by ChEMBL
LigandPNGBDBM50434222(CHEMBL2385487)
Affinity DataKi:  2nMAssay Description:Inhibition of MMP12 (unknown origin)-mediated Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)
Affinity DataKi:  2nMAssay Description:Inhibition of [3H]PDBu binding to PKCepsilon C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206863(CHEMBL3966303)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50206865(CHEMBL3912923)
Affinity DataKi:  2nMAssay Description:Inhibition of recombinant Aurora A kinase derived from human Hela cells using kemptide as substrate in presence of [c-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50115121(CHEMBL3609359)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Human)
Mitsubishi Tanabe Pharma

Curated by ChEMBL
LigandPNGBDBM50343947(2-(6-hydroxy-6-methylheptylamino)-4-methyl-6-(5-me...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  2.90nMAssay Description:Inhibition of [3H]PDBu binding to PKCtheta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187749(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha-1B receptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Rat)
Toray Industries

Curated by ChEMBL
LigandPNGBDBM50187749(3-(1-(3-(piperidin-1-yl)propyl)piperidin-4-yl)-1H-...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosin from alpha1B adrenoceptor in rat liver membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Human)
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)
Affinity DataKi:  3.30nMAssay Description:Inhibition of [3H]PDBu binding to PKCdelta C1B domainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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