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TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.90E+4nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  565nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  6.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  73nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  1.61E+4nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  7.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  75nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB1 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  4.78E+3nMAssay Description:Displacement of 3H-CP-55940 from recombinant full length human CB2 receptor expressed in HEK293 cell membranes after 90 mins by topcount scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  200nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50285610(CHEMBL4170268 | CBV)
Affinity DataEC50:  3.10E+3nMAssay Description:Agonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  6.20E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluorescence as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50061117(6,6,9-Trimethyl-3-pentyl-6H-benzo[c]chromen-1-ol(C...)
Affinity DataEC50:  5.30E+3nMAssay Description:Agonist activity at recombinant rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM20461(Zostrix | (E)-N-[(4-hydroxy-3-methoxyphenyl)methyl...)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50554641(CHEMBL554265)
Affinity DataEC50:  5.40E+3nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50554642(CHEMBL4800169)
Affinity DataEC50:  35nMAssay Description:Agonist activity at human TRPV1 stably transfected in HEK293 cells assessed as increase in calcium influx in presence of ionomycin by Fluo-4-AM dye b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50185034(N-arachidonoyl-O-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataEC50:  250nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50185035(N-arachidonoyl-N-(2-hydroxyethyl)hydroxylamine | C...)
Affinity DataEC50:  260nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50185031(N-oleoyl-N-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataEC50:  400nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM29080(Oleamide MEA | Oleoyl monoethanolamide | CHEMBL280...)
Affinity DataEC50:  890nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50185032(N-palmitoyl-N-(2-hydroxyethyl)hydroxylamine | CHEM...)
Affinity DataEC50:  600nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50185033(N-oleoyl-O-(2-hydroxyethyl)hydroxylamine | CHEMBL2...)
Affinity DataEC50:  320nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM22988(Arachidonoyl ethanolamide | Arachidonoylethanolami...)
Affinity DataEC50:  490nMAssay Description:Agonist activity on human recombinant TRPV1-mediated enhancement of intracellular calcium concentration in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50525957(CHEMBL4461515)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at rat recombinant TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium accumulation by Fluo4-AM based assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622240(CHEMBL5416647)
Affinity DataEC50:  1.88E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622241(CHEMBL5416035)
Affinity DataEC50:  234nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622242(CHEMBL5417721)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622243(CHEMBL5417996)
Affinity DataEC50:  676nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622244(CHEMBL5418018)
Affinity DataEC50:  741nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622245(CHEMBL5403768)
Affinity DataEC50:  841nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622246(CHEMBL5396387)
Affinity DataEC50:  61nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622247(CHEMBL5426686)
Affinity DataEC50:  108nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622248(CHEMBL89848)
Affinity DataEC50:  109nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622249(CHEMBL5428602)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622250(CHEMBL5429923)
Affinity DataEC50:  76nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622251(CHEMBL5422020)
Affinity DataEC50:  7nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622252(CHEMBL5423911)
Affinity DataEC50:  870nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622253(CHEMBL5410131)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622254(CHEMBL5410838)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622255(CHEMBL5423032)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622256(CHEMBL5430219)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622257(CHEMBL5412004)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622258(CHEMBL5417111)
Affinity DataEC50:  37nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622259(CHEMBL5398876)
Affinity DataEC50:  340nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622260(CHEMBL5399027)
Affinity DataEC50:  417nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622261(CHEMBL5432262)
Affinity DataEC50:  586nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622262(CHEMBL5424278)
Affinity DataEC50:  2.44E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM96974(SMR000229037 | cid_836344 | N-benzyl-4-phenylbutan...)
Affinity DataEC50: >5.00E+4nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Eastern Piedmont

Curated by ChEMBL
LigandPNGBDBM50622263(CHEMBL1802306)
Affinity DataEC50:  4.80E+3nMAssay Description:Agonist activity at human recombinant TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM based assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/17/2024
Entry Details
PubMed
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