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TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.15E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.10E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 60nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >2.50E+4nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.45E+3nMAssay Description:Activation of Nrf2 (unknown origin) expressed in human HaCaT-ARE-luc cells after 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.63E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.55E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.63E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.50E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.90E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.62E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.78E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.20E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.28E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 5.00E+3nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.95E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Activation of Nrf2 in human HaCaT-ARE-Luc cells expressing Nqo1 ARE-Luc reporter plasmid incubated for 6 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 7.10E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.14E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 8.90E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 1.14E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 7.10E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: >5.00E+4nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.40E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 2.60E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 6.80E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
TargetEgl nine homolog 1/Prolyl hydroxylase EGLN2/Prolyl hydroxylase EGLN3/Transmembrane prolyl 4-hydroxylase(Human)
University of Eastern Piedmont
Curated by ChEMBL
University of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 5.80E+3nMAssay Description:Inhibition of PHD (unknown origin) expressed in mouse NIH/3T3 cells harboring HRE-driven luciferase gene assessed as transactivation of HIF1alpha aft...More data for this Ligand-Target Pair
