Compile Data Set for Download or QSAR
Found 2252 with Last Name = 'nagase' and Initial = 'h'
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50229232(CHEMBL610527)
Affinity DataKi:  0.00500nMAssay Description:Compound was evaluated for the binding affinity to Opioid receptor mu using [3H]DAMGO as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50229232(CHEMBL610527)
Affinity DataKi:  0.0100nMAssay Description:Compound was evaluated for the binding affinity to opioid receptor kappa using [3H]-EK as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM82552(CAS_111555-58-9 | NTB | naltrindolebenzofuran)
Affinity DataKi:  0.0130nMAssay Description:Compound was evaluated for the binding affinity to opioid receptor delta using [3H]DADLE as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50451343(CHEMBL477154)
Affinity DataKi:  0.0180nMAssay Description:Compound was evaluated for the binding affinity to opioid receptor delta using [3H]DADLE as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50325534(CHEMBL267495 | nalfurafine)
Affinity DataKi:  0.0190nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50596292(CHEMBL5185211)
Affinity DataKi:  0.0272nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50347177(CHEMBL1797687)
Affinity DataKi:  0.0300nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50370067(CHEMBL1237164)
Affinity DataKi:  0.0310nMAssay Description:Compound was evaluated for the binding affinity to opioid receptor delta using [3H]DADLE as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50596293(CHEMBL5188658)
Affinity DataKi:  0.0356nMAssay Description:Displacement of [3H]DPDPE from human KOR expressed in HEK293 cell membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50102826(CHEMBL3339374)
Affinity DataKi:  0.0370nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50491882(CHEMBL3215908)
Affinity DataKi:  0.0370nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50347179(CHEMBL1797689)
Affinity DataKi:  0.0380nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellum homogenate by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50013388(6-Ethyl-3-(1-hydroxy-cyclopropylmethyl)-11,11-dime...)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50102833(CHEMBL3339378)
Affinity DataKi:  0.0430nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50380909(CHEMBL2016678)
Affinity DataKi:  0.0490nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50491882(CHEMBL3215908)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50102826(CHEMBL3339374)
Affinity DataKi:  0.0520nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336669(CHEMBL1672477 | N-[(6beta,14beta-Epoxy-3-hydroxy-1...)
Affinity DataKi:  0.0522nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50229231(CHEMBL610534)
Affinity DataKi:  0.0540nMAssay Description:Compound was evaluated for the binding affinity to opioid receptor delta using [3H]DADLE as radioligand in guinea pig brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50491892(CHEMBL3216338)
Affinity DataKi:  0.0750nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336672(CHEMBL1672473 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.0754nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50491883(CHEMBL3216579)
Affinity DataKi:  0.0810nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336674(CHEMBL1672481 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.0812nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336664((2E)-N-[(17-Cyclopropylmethyl-6beta,14beta-epoxy-3...)
Affinity DataKi:  0.0828nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336677(CHEMBL1672484 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.0833nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336673(CHEMBL1672480 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.0880nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50391602(CHEMBL2147915)
Affinity DataKi:  0.0920nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50380906(CHEMBL2016675)
Affinity DataKi:  0.0970nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50277471((1R,9R,10S,13R)-17-(cyclopropylmethyl)-13-(hydroxy...)
Affinity DataKi:  0.102nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336670(CHEMBL1672478 | N-[(6beta,14beta-Epoxy-3-hydroxy-1...)
Affinity DataKi:  0.108nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336667(CHEMBL1672470 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.109nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50253136(CHEMBL4075409)
Affinity DataKi:  0.109nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain without cerebellum membraneMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50491883(CHEMBL3216579)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50491884(CHEMBL3216801)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50491892(CHEMBL3216338)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50491897(CHEMBL2387739)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in mouse whole brain devoid of cerebellumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50380911(CHEMBL2016680)
Affinity DataKi:  0.110nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50102828(CHEMBL3339372)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336674(CHEMBL1672481 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.110nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Mus musculus (Mouse))
University of Tsukuba

Curated by ChEMBL
LigandPNGBDBM50118178(CHEMBL3613172)
Affinity DataKi:  0.113nMAssay Description:Displacement of [3H]U69,593 from KOR in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336679(CHEMBL1672486 | N-[(6beta,14beta-Epoxy-3-hydroxy-1...)
Affinity DataKi:  0.116nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336667(CHEMBL1672470 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50360146(CHEMBL1929368)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in mouse whole brain membranes without cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336671(CHEMBL1672479 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50102832(CHEMBL3339379)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]U-69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50380911(CHEMBL2016680)
Affinity DataKi:  0.120nMAssay Description:Displacement of [3H]U-69,593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336672(CHEMBL1672473 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.121nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in guinea pig forebrainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336663(2-Phenyl-N-[(17-cyclopropylmethyl-6beta,14beta-epo...)
Affinity DataKi:  0.124nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50336666(CHEMBL1672468 | N-[(17-Cyclopropylmethyl-6beta,14b...)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50599576(CHEMBL5200218)
Affinity DataKi:  0.126nMAssay Description:Displacement of [3H]-DAMGO from recombinant human MOR expressed in CHO cell membranes measured after 2 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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