Report error Found 88 with Last Name = 'nakashima' and Initial = 'm'
Affinity DataEC50: 0.0150nMAssay Description:Agonist activity at human MT1 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0220nMAssay Description:Agonist activity at human MT1 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
Affinity DataEC50: 0.850nMAssay Description:Agonist activity at human MT2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
Affinity DataEC50: 0.530nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0210nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
Affinity DataEC50: 0.820nMAssay Description:Agonist activity at human MT2 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
Affinity DataEC50: 0.0260nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
Affinity DataEC50: 0.510nMAssay Description:Agonist activity at human MT2 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
Affinity DataIC50: 6.40nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 160nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 270nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 730nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+3nMAssay Description:Antagonist activity at OX1R intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at OX1R intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+3nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.70E+3nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.40E+3nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.20E+3nMAssay Description:Antagonist activity at human OX2R expressed in CHO cells assessed intracellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.00650nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.00820nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0140nMAssay Description:Binding affinity to human MT1 expressed in CHO cellsMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 0.0260nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0270nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT1 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0310nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT1 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0370nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT1 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0390nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0440nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0580nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0620nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT1 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT1 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0730nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0820nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0830nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0850nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.0860nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0880nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.112nMAssay Description:Binding affinity to human MT2 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Displacement of 2-[125I]iodomelatonin from human MT2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Displacement of 2-[125l]-lodomelatonin from human MT2 expressed in CHO cell membrane incubated for 150 mins by radioligand binding assayMore data for this Ligand-Target Pair
