Compile Data Set for Download or QSAR
Found 108 with Last Name = 'nardone' and Initial = 'na'
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218166((R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataKi:  10nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218173((R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  21nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218170((R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  30nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218180((R)-2-(2-(4-(2-ethylthiazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218168((R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino...)
Affinity DataKi:  37nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218167((R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethyla...)
Affinity DataKi:  49nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218177((R)-2-(2-(4-(2-(benzyloxymethyl)oxazol-4-yl)phenox...)
Affinity DataKi:  50nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218176((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-4-yl)thia...)
Affinity DataKi:  97nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218182((R)-1-(pyridin-3-yl)-2-(2-(4-(2-(trifluoromethyl)t...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218164((R)-2-(2-(4-(2-methylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218185((1R)-1-(pyridin-3-yl)-2-(2-(4-(2-(pyridin-3-yl)thi...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218172((R)-2-(2-(4-(2-cyclopentylthiazol-4-yl)phenoxy)eth...)
Affinity DataKi:  130nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218165((R)-1-(pyridin-3-yl)-2-(2-(4-(thiazol-4-yl)phenoxy...)
Affinity DataKi:  140nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218174((R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  150nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218181((R)-2-(2-(4-(5-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  170nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218166((R)-2-(2-(4-(oxazol-4-yl)phenoxy)ethylamino)-1-(py...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218171((R)-2-(2-(4-(2-(methoxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218170((R)-2-(2-(4-(2-(hydroxymethyl)oxazol-4-yl)phenoxy)...)
Affinity DataKi:  270nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218167((R)-2-(2-(4-(2-isopropyloxazol-4-yl)phenoxy)ethyla...)
Affinity DataKi:  360nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218173((R)-2-(2-(4-(2-methyloxazol-4-yl)phenoxy)ethylamin...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218168((R)-2-(2-(4-(2-ethyloxazol-4-yl)phenoxy)ethylamino...)
Affinity DataKi:  400nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218174((R)-2-(2-(4-(2-phenylthiazol-4-yl)phenoxy)ethylami...)
Affinity DataKi:  500nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50218179((R)-2-(2-(4-(2,5-dimethyloxazol-4-yl)phenoxy)ethyl...)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [125I]iodocyanopindolol from human adrenergic beta-1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329182(CHEMBL1269261 | N-benzyl-N-isopropyl-2-(5-oxo-1-ph...)
Affinity DataIC50:  2nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329179(2-((4S)-4-((1H-indol-3-yl)methyl)-5-oxo-1-phenyl-4...)
Affinity DataIC50:  12.2nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329184(CHEMBL1269262 | N-benzyl-N-isopropyl-2-(5-oxo-4-ph...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329180(3-((6-(2-(isopropyl(phenyl)amino)-2-oxoethyl)-5-ox...)
Affinity DataIC50:  19.7nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329185(2-(4-(1H-indazol-3-yl)-5-oxo-1-phenyl-4H-benzo[b][...)
Affinity DataIC50:  21nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329182(CHEMBL1269261 | N-benzyl-N-isopropyl-2-(5-oxo-1-ph...)
Affinity DataIC50:  24.3nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329179(2-((4S)-4-((1H-indol-3-yl)methyl)-5-oxo-1-phenyl-4...)
Affinity DataIC50:  31.7nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329185(2-(4-(1H-indazol-3-yl)-5-oxo-1-phenyl-4H-benzo[b][...)
Affinity DataIC50:  48.5nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329181(3-(6-(2-(benzyl(isopropyl)amino)-2-oxoethyl)-5-oxo...)
Affinity DataIC50:  49.3nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(RAT)
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataIC50:  52.6nMAssay Description:Displacement of [125I]CCK8 from rat CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329178((S)-3-(3-(1-(2-(isopropyl(phenyl)amino)-2-oxoethyl...)
Affinity DataIC50:  131nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329183(2-(4-benzyl-5-oxo-1-phenyl-4H-benzo[b][1,2,4]triaz...)
Affinity DataIC50:  201nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50329186(2-((4R)-4-(1H-indol-3-yl)-5-oxo-1-phenyl-4H-benzo[...)
Affinity DataIC50:  246nMAssay Description:Displacement of [125I]CCK8 from human CCK1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147439((2R,6S)-2,6-Dimethyl-morpholine-4-sulfonic acid {4...)
Affinity DataEC50:  8nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147440(CHEMBL542928 | N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-...)
Affinity DataEC50:  165nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147441(4-Phenyl-piperidine-1-sulfonic acid {4-[2-((R)-2-h...)
Affinity DataEC50:  47nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147442(4-Methyl-piperazine-1-sulfonic acid {4-[2-((R)-2-h...)
Affinity DataEC50:  41nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147444(CHEMBL553279 | N-[4-(2-{[(2R)-2-hydroxy-2-pyridin-...)
Affinity DataEC50:  7nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147443(CHEMBL110969 | N'-[4-(2-{[(2R)-2-(3-chlorophenyl)-...)
Affinity DataEC50:  537nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147447(CHEMBL556022 | Piperidine-1-sulfonic acid {4-[2-((...)
Affinity DataEC50:  99nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147445(CHEMBL544338 | N'-[4-(2-{[(2R)-2-hydroxy-2-pyridin...)
Affinity DataEC50:  943nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147446(4-Methyl-piperidine-1-sulfonic acid {4-[2-((R)-2-h...)
Affinity DataEC50:  36nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50147448(4-Phenyl-piperidine-1-sulfonic acid {4-[2-((R)-2-h...)
Affinity DataEC50:  23nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Pfizer Inc

Curated by ChEMBL
LigandPNGBDBM50092645((R)-N-(4-(2-(2-hydroxy-2-(pyridin-3-yl)ethylamino)...)
Affinity DataEC50:  3nMAssay Description:Agonist activity (EC50) was assessed by measuring cAMP levels in CHO cells expressing cloned human Beta-3 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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