Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 104 with Last Name = 'norcini' and Initial = 'g'
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of human VCAM and Ramos cell VLA-4 interactionMore data for this Ligand-Target Pair
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataKi:  1.5nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human VCAM and Ramos cell VLA-4 interactionMore data for this Ligand-Target Pair
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM14361((R,S)-Rolipram | 4-(3-cyclopentyloxy-4-methoxy-phe...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
LigandPNGBDBM50219407(CHEMBL84350)
Affinity DataKi:  5nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218261(CHEMBL74631)
Affinity DataKi:  13nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218265(CHEMBL308407)
Affinity DataKi:  16nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218578(CHEMBL79902)
Affinity DataKi:  17nMAssay Description:Affinity for alpha4-beta1 integrin from HL60 cell lysateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218586(CHEMBL79471)
Affinity DataKi:  34nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataKi:  38nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
LigandPNGBDBM50346088((1r,4r)-4-cyano-4-(3-(cyclopentyloxy)-4-methoxyphe...)
Affinity DataKi:  38nMAssay Description:Inhibition of rolipram binding to Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM50218262(CHEMBL308158)
Affinity DataKi:  46nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219414(CHEMBL79661)
Affinity DataKi:  60nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219411(CHEMBL82934)
Affinity DataKi:  63nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218267(CHEMBL74404)
Affinity DataKi:  71nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218589(CHEMBL79535)
Affinity DataKi:  89nMAssay Description:Inhibition of alpha4-beta1 VCAM binding in Jurkat cell adhesion assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50092350((5-Cyclopentyloxy-6-methoxy-phthalazin-1-yl)-(3,5-...)
Affinity DataKi:  95nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218264(CHEMBL72362)
Affinity DataKi:  121nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219417(CHEMBL421343)
Affinity DataKi:  128nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219409(CHEMBL354743)
Affinity DataKi:  138nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataKi:  149nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataKi:  149nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218260(CHEMBL70391)
Affinity DataKi:  149nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218268(CHEMBL309341)
Affinity DataKi:  164nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219404(CHEMBL79739)
Affinity DataKi:  199nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218588(CHEMBL312375)
Affinity DataKi:  204nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219406(CHEMBL309420)
Affinity DataKi:  208nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219413(CHEMBL81226)
Affinity DataKi:  212nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219405(CHEMBL81020)
Affinity DataKi:  235nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219410(CHEMBL311025)
Affinity DataKi:  237nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218580(CHEMBL310387)
Affinity DataKi:  271nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218269(CHEMBL73640)
Affinity DataKi:  286nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218263(CHEMBL419814)
Affinity DataKi:  320nMAssay Description:Inhibition of rolipram binding to PDE4 from human neutrophilsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218583(CHEMBL81364)
Affinity DataKi:  383nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219408(CHEMBL84115)
Affinity DataKi:  397nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218587(CHEMBL312322)
Affinity DataKi:  436nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218585(CHEMBL3085289)
Affinity DataKi:  452nMAssay Description:Inhibition of rolipram binding to PDE4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219416(CHEMBL167389)
Affinity DataKi:  473nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219412(CHEMBL82882)
Affinity DataKi:  498nMAssay Description:Affinity for rolipram binding site (RBS) of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human Phosphodiesterase 4More data for this Ligand-Target Pair
LigandPNGBDBM14775(3-(cyclopentyloxy)-N-(3,5-dichloropyridin-4-yl)-4-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of Phosphodiesterase 4 from human neutrophilsMore data for this Ligand-Target Pair
TargetNeprilysin(Rat)
R & D, Zambon Group

LigandPNGBDBM85431(NEP inhibitor, 6k)
Affinity DataIC50:  2nMT: 25°CAssay Description:Enzyme inhibition assay using neutrol endopeptiase EC 3.4.24.11 (NEP).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rat)
R & D, Zambon Group

LigandPNGBDBM85433(NEP inhibitor, 6m)
Affinity DataIC50:  2nMT: 25°CAssay Description:Enzyme inhibition assay using neutrol endopeptiase EC 3.4.24.11 (NEP).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rat)
R & D, Zambon Group

LigandPNGBDBM85434(NEP inhibitor, 6n)
Affinity DataIC50:  2nMT: 25°CAssay Description:Enzyme inhibition assay using neutrol endopeptiase EC 3.4.24.11 (NEP).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50219407(CHEMBL84350)
Affinity DataIC50:  2nMAssay Description:Inhibition of human neutrophil phosphodiesterase type IV (PDE4)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Rat)
R & D, Zambon Group

LigandPNGBDBM85429(NEP inhibitor, 6i)
Affinity DataIC50:  3nMT: 25°CAssay Description:Enzyme inhibition assay using neutrol endopeptiase EC 3.4.24.11 (NEP).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218578(CHEMBL79902)
Affinity DataIC50:  4nMAssay Description:Inhibition of human Phosphodiesterase 4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50218582(CHEMBL123993)
Affinity DataIC50:  4nMAssay Description:Inhibition of human VCAM binding to VLA-4 of Ramos cells in ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 104 total ) | Next | Last >>
Jump to: