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TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186366(c(his-L-phe-arg-trp-Aoc) | CHEMBL211131)
Affinity DataEC50:  5.10E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186366(c(his-L-phe-arg-trp-Aoc) | CHEMBL211131)
Affinity DataEC50:  9.59E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186368(c(his-D-phe-arg-trp-Abu) | CHEMBL379531)
Affinity DataEC50:  270nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186369(c(his-D-phe-arg-trp-Ava) | CHEMBL210399)
Affinity DataEC50:  1.01E+4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  1.80nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186371(c(his-D-phe-arg-trp-Aoc) | CHEMBL264120)
Affinity DataEC50:  16.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186369(c(his-D-phe-arg-trp-Ava) | CHEMBL210399)
Affinity DataEC50:  3.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186372(c(his-D-phe-arg-trp-betaala) | CHEMBL380198)
Affinity DataEC50:  135nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(c(his-D-phe-arg-trp-Ahp) | CHEMBL379959)
Affinity DataEC50:  15.4nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186372(c(his-D-phe-arg-trp-betaala) | CHEMBL380198)
Affinity DataEC50:  1.11E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186368(c(his-D-phe-arg-trp-Abu) | CHEMBL379531)
Affinity DataEC50:  1.58E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186370(c(his-D-phe-arg-trp-Ahx) | CHEMBL379627)
Affinity DataEC50:  1.30E+3nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  72.9nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186370(c(his-D-phe-arg-trp-Ahx) | CHEMBL379627)
Affinity DataEC50:  3.12E+3nMAssay Description:Activity at human MC4R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186367(c(his-D-phe-arg-trp-Ahp) | CHEMBL379959)
Affinity DataEC50:  67nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetMelanocyte-stimulating hormone receptor(Human)
Asahi Kasei Pharma

Curated by ChEMBL
LigandPNGBDBM50186371(c(his-D-phe-arg-trp-Aoc) | CHEMBL264120)
Affinity DataEC50:  77.4nMAssay Description:Activity at human MC1R by cAMP accumulation in SaoS2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50378580(CHEMBL437430)
Affinity DataEC50:  1.09nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304252((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  6.94nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304253((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  8.51nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304254((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  12.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304255((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  13.2nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304256((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  10.1nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304257((6S,9S,12S,15S,20aS)-9-((1H-indol-3-yl)methyl)-12-...)
Affinity DataEC50:  75.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304258((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  20.6nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetUrotensin-2 receptor(Human)
Prism Bio. Lab.

Curated by ChEMBL
LigandPNGBDBM50304259((6S,9S,12S,15S,20aS)-9,15-bis((1H-indol-3-yl)methy...)
Affinity DataEC50:  16.7nMAssay Description:Agonist activity at human GPR14 expressed in HEK293 cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50292220(1-[2-[(S)-(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-ph...)
Affinity DataIC50: 0.0710nMAssay Description:Inhibitory concentration in guinea-pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212609(Dmt-Pro-Dmp-Phe-NH2 | CHEMBL228409)
Affinity DataIC50: 0.120nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212608(Dmt-Pro-Mmp-Phe-NH2 | CHEMBL389948)
Affinity DataIC50: 0.160nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212617(Dmt-Pro-Emp-Phe-NH2 | CHEMBL374818)
Affinity DataIC50: 0.170nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063918((2R,3S)-N*4*-Hydroxy-2-isobutyl-N*1*-((S)-1-methyl...)
Affinity DataIC50: 0.200nMAssay Description:Activity against Matrix metalloprotease-9 (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063912((R)-N*4*-Hydroxy-N*1*-((S)-methylcarbamoyl-phenyl-...)
Affinity DataIC50: 0.200nMAssay Description:Activity against Matrix metalloprotease-9 (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212618(Dmt-Pro-Imp-Phe-NH2 | CHEMBL228516)
Affinity DataIC50: 0.200nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212621(Dmt-Pro-Tmp-Phe-NH2 | CHEMBL228503)
Affinity DataIC50: 0.210nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50: 0.260nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataIC50: 0.261nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 0.270nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig intestine assessed as inhibition of electrically evoked myenteric plexus longitudinal mu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063915((2R,3S)-N*4*-Hydroxy-2-isobutyl-3-methyl-N*1*-[(S)...)
Affinity DataIC50: 0.300nMAssay Description:Activity against Matrix metalloprotease-9 (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063915((2R,3S)-N*4*-Hydroxy-2-isobutyl-3-methyl-N*1*-[(S)...)
Affinity DataIC50: 0.300nMAssay Description:Activity against Matrix metalloprotease-2 (MMP-2).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063915((2R,3S)-N*4*-Hydroxy-2-isobutyl-3-methyl-N*1*-[(S)...)
Affinity DataIC50: 0.300nMAssay Description:Activity against Matrix metalloprotease-1 (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50272031((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 0.320nMAssay Description:Agonist activity at mu opioid receptor in human SHSY5Y cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212613(Tyr-Pro-Dmp-Phe-NH2 | CHEMBL266122)
Affinity DataIC50: 0.380nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetInterstitial collagenase(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063918((2R,3S)-N*4*-Hydroxy-2-isobutyl-N*1*-((S)-1-methyl...)
Affinity DataIC50: 0.400nMAssay Description:Activity against Matrix metalloprotease-1 (MMP-1).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
University of Queensland

Curated by ChEMBL
LigandPNGBDBM50199865((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...)
Affinity DataIC50: 0.430nMAssay Description:Agonist activity at mu opioid receptor in human SHSY5Y cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetMatrix metalloproteinase-9(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.5nMAssay Description:Activity against Matrix metalloprotease-9 (MMP-9).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50172014(H-Dmt-D-Arg(NO2)-Phe-Lys(Z)-NH2 | CHEMBL371856)
Affinity DataIC50: 0.509nMAssay Description:Agonist activity against mu opioid receptor of guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50212617(Dmt-Pro-Emp-Phe-NH2 | CHEMBL374818)
Affinity DataIC50: 0.510nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159685(5N-[1-[1-carbamoyl-2-phenyl-(1S)-ethylcarbamoyl]-2...)
Affinity DataIC50: 0.590nMAssay Description:In vitro inhibition of opioid receptor delta using mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50149384((S)-1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...)
Affinity DataIC50: 0.590nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferens assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetStromelysin-1(Human)
Kanebo

Curated by ChEMBL
LigandPNGBDBM50063915((2R,3S)-N*4*-Hydroxy-2-isobutyl-3-methyl-N*1*-[(S)...)
Affinity DataIC50: 0.600nMAssay Description:Activity against Matrix metalloprotease-3 (MMP-3).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50159681((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...)
Affinity DataIC50: 0.623nMAssay Description:In vitro inhibition of opioid receptor mu using isolated guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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